Title:
殺虫特性を有する4’-及び4”-位において置換されたエバーメクチン及びエバーメクチンモノサッカライド
Document Type and Number:
Japanese Patent JP4908213
Kind Code:
B2
Abstract:
Described is a compound of the formula (I) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and either (A) R2 is —N(R3)R4, and (1) X is 0, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl; or (2) X is S, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl; or (3) X is 0 or S, wherein R3 and R4 together are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) R2 is OR5, X is 0 or S, wherein R5 is, for instance, C1-C12alkyl, mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity.
Inventors:
Murphy Quesavi, Fiona
Pittelna, Thomas
Myenfish, Peter
Cassel, Jerome
Caranta, Laura
June, Pierre
Fetter, Ottomar Franz
Pittelna, Thomas
Myenfish, Peter
Cassel, Jerome
Caranta, Laura
June, Pierre
Fetter, Ottomar Franz
Application Number:
JP2006524341A
Publication Date:
April 04, 2012
Filing Date:
August 27, 2004
Export Citation:
Assignee:
Merial Limited
International Classes:
C07H17/08; A01N43/90; A01P7/04; C07H19/01
Domestic Patent References:
| JP7500844A | ||||
| JP2078683A | ||||
| JP54061197A | ||||
| JP2264778A | ||||
| JP2212491A |
Foreign References:
| US4833168 |
Other References:
MROZIK,H. et al,Avermectin acyl derivatives with anthelmintic activity,Journal of Medicinal Chemistry,1982年,Vol.25, No.6,pp.658-663
Attorney, Agent or Firm:
Atsushi Aoki
Takashi Ishida
Fukumoto product
Tetsuji Koga
Yoichi Watanabe
Masaru Nakajima
Tatsunori Ikeda
Takashi Ishida
Fukumoto product
Tetsuji Koga
Yoichi Watanabe
Masaru Nakajima
Tatsunori Ikeda