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Title:
ニューロキニンアンタゴニストを含む製剤
Document Type and Number:
Japanese Patent JP2010513356
Kind Code:
A
Abstract:
Pharmaceutical compositions in the form of a solid dispersion comprising (4R)-4-[N'-methyl-N'-(3,5-bistrifluoromethyl-benzoyl)-amino]-4-(3,4-dichlorobenzyl)-but-2-enoic acid N-[(R)-cpsilon-caprolactam-3-yl]-amidc or a pharmaceutically acceptable salt or solvate thereof and a carrier. Such compositions are useful to treat patients who have functional motility disorders of the viscera, especially irritable bowel syndrome or functional dyspepsia, or urinary bladder disorders, especially urinary incontinence.

Inventors:
Anke Diederich
Carsten Timpe
Angelica Reese
Isabelle Ottinger
Irene Mueller
Michael Herbig
Helmut Schutz
Jay Pershban Lakshman
Oscar Culp
Application Number:
JP2009541897A
Publication Date:
April 30, 2010
Filing Date:
December 20, 2007
Export Citation:
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Assignee:
Novartis Age
International Classes:
A61K31/55; A61K9/10; A61K9/14; A61K9/20; A61K47/04; A61K47/12; A61K47/26; A61K47/32; A61K47/36; A61K47/38; A61P1/04; A61P1/12; A61P1/14; A61P11/00; A61P11/06; A61P13/02; A61P13/10
Domestic Patent References:
JP2008536913A2008-09-11
JP2001521899A2001-11-13
JP2007509184A2007-04-12
JP2007520521A2007-07-26
JP2001503387A2001-03-13
JP2003526666A2003-09-09
JPH054919A1993-01-14
JP2004131393A2004-04-30
Foreign References:
WO2005039563A22005-05-06
WO2005074891A12005-08-18
WO2006112649A12006-10-26
Attorney, Agent or Firm:
Mitsuo Tanaka
Takuji Yamada
Mitsutaka Iwasaki
Aoyama Aoi
Masayuki Nakagawa