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Title:
フマル酸エステルのプロドラッグおよび種々の疾患の治療におけるその使用
Document Type and Number:
Japanese Patent JP6587648
Kind Code:
B2
Abstract:
The present invention provides compounds of formula (I), and pharmaceutical compositions thereof.

Inventors:
Zeidan, Tarek, A.
Duncan, Scott
Henken, Christopher, Pee.
Win, Thomas, Andrew
Sanreme, Carlos, N.
Application Number:
JP2017070509A
Publication Date:
October 09, 2019
Filing Date:
March 31, 2017
Export Citation:
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Assignee:
Arcames Pharma Ireland Limited
International Classes:
C07C219/08; A61K31/155; A61K31/221; A61K31/222; A61K31/36; A61K31/40; A61K31/4015; A61K31/41; A61K31/415; A61K31/4164; A61K31/4166; A61K31/4184; A61K31/4192; A61K31/4196; A61K31/421; A61K31/426; A61K31/44; A61K31/4402; A61K31/4409; A61K31/4425; A61K31/445; A61K31/495; A61K31/505; A61K31/519; A61K31/5375; A61K31/5383; A61K31/54; A61K31/55; A61P25/00; C07C229/06; C07C233/17; C07C243/38; C07C271/10; C07C275/06; C07C279/08; C07C317/18; C07C327/48; C07C333/20; C07C335/16; C07C337/06; C07D207/325; C07D207/34; C07D207/408; C07D207/448; C07D209/08; C07D211/40; C07D211/44; C07D213/64; C07D213/74; C07D213/81; C07D213/85; C07D213/89; C07D231/12; C07D233/34; C07D233/42; C07D233/61; C07D233/74; C07D235/08; C07D239/36; C07D239/54; C07D239/88; C07D239/96; C07D249/04; C07D249/08; C07D257/04; C07D263/04; C07D263/24; C07D265/30; C07D265/32; C07D277/42; C07D279/12; C07D295/088; C07D295/15; C07D295/24; C07D317/66; C07D498/08
Domestic Patent References:
JP2012500285A
JP2011231094A
JP2009510137A
JP2000513023A
JP2214731A
JP62199643A
Foreign References:
EP0928820A1
US3892671
WO2012014162A1
WO2011085211A1
WO2013119791A1
WO2013181451A1
WO2014031844A1
WO2014031892A1
Other References:
Biochimica et Biophysica Acta, Protein Structure and Molecular Enzymology,1986年,870(2),p.357-366
Chemical Communications (Cambridge, United Kingdom) ,2010年,46(42),p.7993-7995,Supplementary Information p.1-30
Journal of Organic Chemistry,1993年,58(24),p.6745-6755
Acta Polymerica,1982年,33(3),p.215-217
Naunyn-Schmiedebergs Archiv fuer Experimentelle Pathologie und Pharmakologie,1955年,225,p.541-50
Attorney, Agent or Firm:
Yoshinori Hosoda