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Patent Searching and Data


Title:
縮合二環式化合物、その組成物及び応用
Document Type and Number:
Japanese Patent JP7301758
Kind Code:
B2
Abstract:
Fused bicyclic compounds are inhibitors of GPR91. The compounds, their stereoisomers, tautomers, prodrugs, polymorphs, solvates, pharmaceutically acceptable salts, and pharmaceutical compositions containing them are useful in the treatment, prevention, prophylaxis, management, or adjunct treatment of all medical conditions related to inhibition of GPR91.

Inventors:
Nadim Shaikh
Mahesh Tukkar
Shiresh Cinde
Manoji Joshi
Keshav Nike
Amit Valerao
Mayur Mukim
Devnath Bunya
B-Mashankar-Kurkarni
Qasim Mooktial
Application Number:
JP2019571826A
Publication Date:
July 03, 2023
Filing Date:
March 13, 2018
Export Citation:
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Assignee:
IMPETIS BIOSCIENCES LIMITED
International Classes:
C07D217/02; A61K31/357; A61K31/404; A61K31/405; A61K31/416; A61K31/4184; A61K31/4192; A61K31/437; A61K31/472; A61K31/4725; A61K31/502; A61K31/517; A61K45/00; A61P1/16; A61P3/00; A61P9/00; A61P9/12; A61P13/12; A61P27/02; A61P29/00; A61P35/00; C07C57/62; C07D209/08; C07D215/06; C07D215/233; C07D217/04; C07D217/26; C07D231/56; C07D237/30; C07D239/74; C07D265/36; C07D319/18; C07D401/12; C07D471/04
Domestic Patent References:
JP2003528871A
JP2014520885A
JP58021672A
Foreign References:
WO1997025321A2
Other References:
Bioorganic & Medicinal Chemistry Letters,2011年,Vol.21,pp.3596-3602
Chemical Abstract,89:146562,Retrieved from STN international [online] ;retrieved on 2 March 2022
Database REGISTRY,2011年,RN 1348552-37-3, 904281-92-1, 904034-97-5, 330561-55-2, 328265-88-9, 328265-86-7, 328265-73-2, 328265-40-3, 313530-69-7, 312759-09-4, 297743-29-4, 294890-77-0,Retrieved from STN international [online] ;retrieved on 2 March 2022
Attorney, Agent or Firm:
Norito Yamao
Sei Morimoto
Yasushi Ochiai