Title:
グルココルチコイド受容体モジュレーター
Document Type and Number:
Japanese Patent JP3901945
Kind Code:
B2
Abstract:
The present invention provides non-steroidal compounds of formula I which are selective modulators (i.e., agonist and antagonists) of a steroid receptor, specifically, the glucocorticoid receptor. The present invention also provides pharmaceutical compositions containing these compounds and methods for using these compounds to treat animals requiring glucocorticoid receptor agonist or antagonist therapy. Glucocorticoid receptor modulators are useful to treat diseases, such as obesity, diabetes, inflammation and others as described below. The present invention also provides intermediates and processes for preparing these compounds
Inventors:
Dow, Robert Lee
Ryu, Kevin Khun-Chin
Bradley Paul, Morgan
Andrew Gordon, Swick
Ryu, Kevin Khun-Chin
Bradley Paul, Morgan
Andrew Gordon, Swick
Application Number:
JP2000615356A
Publication Date:
April 04, 2007
Filing Date:
March 27, 2000
Export Citation:
Assignee:
Pfizer Products Inc.
International Classes:
C07C49/755; A61K31/05; C07D295/12; A61K31/122; A61K31/27; A61K31/275; A61K31/325; A61K31/40; A61K31/4164; A61K31/44; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4965; A61K31/5375; A61P3/04; A61P3/10; A61P11/06; A61P19/02; A61P25/22; A61P25/24; A61P25/28; A61P27/16; A61P29/00; A61P37/02; A61P43/00; C07C35/42; C07C49/675; C07C49/737; C07C49/747; C07C49/757; C07C65/17; C07C69/00; C07C215/50; C07C215/74; C07C225/22; C07C233/58; C07C235/48; C07C235/66; C07C247/24; C07C251/44; C07C251/52; C07C251/60; C07C255/53; C07C255/54; C07C271/10; C07C271/44; C07C271/52; C07C281/04; C07C307/02; C07C309/65; C07C309/66; C07C309/73; C07C311/04; C07C311/08; C07C311/51; C07C317/18; C07C333/04; C07D207/09; C07D211/46; C07D213/22; C07D213/30; C07D213/40; C07D213/75; C07D231/40; C07D231/56; C07D233/61; C07D239/34; C07D241/12; C07D241/18; C07D241/20; C07D249/08; C07D249/14; C07D257/04; C07D271/06; C07D271/07; C07D277/24; C07D277/28; C07D277/56; C07D295/092; C07D295/13; C07D295/185; C07D295/205; C07D303/14; C07D317/36; C07D333/16; C07D413/04; C07D455/06
Domestic Patent References:
| JP61271216A | ||||
| JP62056422A | ||||
| JP61083138A | ||||
| JP45011139B1 |
Foreign References:
| US5039706 | ||||
| US3516993 |
Other References:
Int. J. Biochem.,1989年,21(5),p.463-468
Journal of Chemical Society, Perkin Transactions I,1982年,(1),p.201-204
Tetrahedron,1995年,51(33),p.9079-9090
Tetrahedron Letters,1986年,27(33),p.3913-3914
Tetrahedron Letters,1986年,27(38),p.4541-4544
Journal of the American Chemical Society,1965年,87(1),p.82-86
Tetrahedron,1994年,50(19),p.5645-5658
Heterocycles,1994年,37(1),p.303-309
Journal of Chemical Society, Perkin Transactions I,1982年,(1),p.201-204
Tetrahedron,1995年,51(33),p.9079-9090
Tetrahedron Letters,1986年,27(33),p.3913-3914
Tetrahedron Letters,1986年,27(38),p.4541-4544
Journal of the American Chemical Society,1965年,87(1),p.82-86
Tetrahedron,1994年,50(19),p.5645-5658
Heterocycles,1994年,37(1),p.303-309
Attorney, Agent or Firm:
Kazuo Shamoto
Shosuke Imai
Tadashi Masui
Yasushi Kobayashi
Hiroyuki Tomita
Tadahiko Kurita
Shosuke Imai
Tadashi Masui
Yasushi Kobayashi
Hiroyuki Tomita
Tadahiko Kurita
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