Title:
配糖体含有リポソーム
Document Type and Number:
Japanese Patent JP4728805
Kind Code:
B2
Abstract:
A drug product which can maximize the effect of a cholestanol glycoside useful as an anticancer agent. The present invention provides a liposomal composition containing a glycoside exhibiting antitumor activity, a phospholipid, and a positive-charge-providing substance; the glycoside being composed of GlcNAc-Gal-, GlcNAc-Gal-Glc-, Fuc-Gal-, Gal-Glc-, or Gal- as a sugar moiety, and a hydrophobic compound capable of forming a liposome.
Inventors:
Yazawa Shin
Izumi Takai
Nishimura Toyo
Izumi Takai
Nishimura Toyo
Application Number:
JP2005511840A
Publication Date:
July 20, 2011
Filing Date:
July 15, 2004
Export Citation:
Assignee:
Otsuka Pharmaceutical Co., Ltd.
International Classes:
A61K31/704; A61K9/127; A61K31/7032; A61K47/18; A61K47/24; A61P35/00; C07H15/10; C07H15/18; C07J17/00
Domestic Patent References:
JPH1160592A | 1999-03-02 | |||
JP2000191685A | 2000-07-11 | |||
JPH03279394A | 1991-12-10 | |||
JPH0193562A | 1989-04-12 | |||
JP2002503685A | 2002-02-05 | |||
JP2000319200A | 2000-11-21 | |||
JP2001354639A | 2001-12-25 |
Attorney, Agent or Firm:
Alga Patent Office, a patent business corporation
Miyuki Ariga
Toshio Takano
Toshio Nakajima
Masaki Murata
Hiroto Yamamoto
Miyuki Ariga
Toshio Takano
Toshio Nakajima
Masaki Murata
Hiroto Yamamoto