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Title:
ヘテロアリール置換ピペラジニル-ピリジン類縁体
Document Type and Number:
Japanese Patent JP2008528506
Kind Code:
A
Abstract:
Substituted biaryl piperazinyl-pyridine analogues are provided, of the Formula: wherein variables are as described herein. Such compounds are ligands that may be used to modulate specific receptor activity in vivo or in vitro, and are particularly useful in the treatment of conditions associated with pathological receptor activation in humans, domesticated companion animals and livestock animals. Pharmaceutical compositions and methods for using such compounds to treat such disorders are provided, as are methods for using such ligands for receptor localization studies.

Inventors:
Charles A Bloom
Application Number:
JP2007552316A
Publication Date:
July 31, 2008
Filing Date:
January 19, 2006
Export Citation:
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Assignee:
Neurogen Corporation
International Classes:
C07D401/14; A61K31/506; A61K31/5377; A61P3/04; A61P11/00; A61P11/06; A61P13/02; A61P13/10; A61P17/04; A61P25/04; A61P43/00; C07D403/14; C07D413/14; C07D417/14; G01N33/15; G01N33/50; G01N33/543
Attorney, Agent or Firm:
Norio Saeki