Title:
前立腺がんの内部放射線療法のための前立腺特異的膜抗原を標的とした高親和性薬剤
Document Type and Number:
Japanese Patent JP7073270
Kind Code:
B2
Abstract:
Prostate-specific membrane antigen targeted high-affinity agents for endoradiotherapy of prostate cancer are disclosed.
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Inventors:
Sangita Ray
Martin Gee Pumper
Martin Gee Pumper
Application Number:
JP2018549808A
Publication Date:
May 23, 2022
Filing Date:
March 22, 2017
Export Citation:
Assignee:
The Johns Hopkins University
International Classes:
C07D257/02; C07D401/12
Domestic Patent References:
| JP2014524419A |
Foreign References:
| WO2017116994A1 | ||||
| WO2015055318A1 | ||||
| WO2015171792A1 | ||||
| WO2013082338A1 | ||||
| WO2010065902A1 | ||||
| WO2016030329A1 |
Other References:
Eder, Matthias; Schaefer, Martin; Bauder-Wuest, Ulrike; Hull, William-Edmund; Waengler, Carmen; Mier, Walter; Haberkorn, Uwe; Eisenhut, Michael,68Ga-Complex Lipophilicity and the Targeting Property of a Urea-Based PSMA Inhibitor for PET Imaging,Bioconjugate Chemistry,2012年,23(4),,688-697
Benesova, Martina; Bauder-Wuest, Ulrike; Schaefer, Martin; Klika, Karel D.; Mier, Walter; Haberkorn, Uwe; Kopka, Klaus; Eder, Matthias,Linker Modification Strategies To Control the Prostate-Specific Membrane Antigen (PSMA)-Targeting and Pharmacokinetic Properties of DOTA-Conjugated PSMA Inhibitors,Journal of Medicinal Chemistry,2016年,59(5),,1761-1775
Shallal, Hassan M.; Minn, Il; Banerjee, Sangeeta R.; Lisok, Ala; Mease, Ronnie C.; Pomper, Martin G.,Heterobivalent Agents Targeting PSMA and Integrin-αvβ3,Bioconjugate Chemistry,2014年,25(2),,393-405
Banerjee, Sangeeta R.; et al,Synthesis and Evaluation of Technetium-99m- and Rhenium-Labeled Inhibitors of the Prostate-Specific Membrane Antigen (PSMA),Journal of Medicinal Chemistry ,2008年,51(15),,4504-4517
Cleeren, Frederik; Lecina, Joan; Billaud, Emilie M. F.; Ahamed, Muneer; Verbruggen, Alfons; Bormans, Guy M.,New Chelators for Low Temperature Al18F-Labeling of Biomolecules,Bioconjugate Chemistry,2016年,27(3),,790-798
Banerjee, Sangeeta Ray; et al,Synthesis and Evaluation of GdIII-Based Magnetic Resonance Contrast Agents for Molecular Imaging of Prostate-Specific Membrane Antigen,Angewandte Chemie, International Edition,2015年,54(37),,10778-10782
Schaefer, Martin; Bauder-Wuest, Ulrike; Leotta, Karin; Zoller, Frederic; Mier, Walter; Haberkorn, Uwe; Eisenhut, Michael; Eder, Matthias,A dimerized urea-based inhibitor of the prostate-specific membrane antigen for 68Ga-PET imaging of prostate cancer,EJNMMI Research,2012年,2(1),,23
Benesova, Martina; Bauder-Wuest, Ulrike; Schaefer, Martin; Klika, Karel D.; Mier, Walter; Haberkorn, Uwe; Kopka, Klaus; Eder, Matthias,Linker Modification Strategies To Control the Prostate-Specific Membrane Antigen (PSMA)-Targeting and Pharmacokinetic Properties of DOTA-Conjugated PSMA Inhibitors,Journal of Medicinal Chemistry,2016年,59(5),,1761-1775
Shallal, Hassan M.; Minn, Il; Banerjee, Sangeeta R.; Lisok, Ala; Mease, Ronnie C.; Pomper, Martin G.,Heterobivalent Agents Targeting PSMA and Integrin-αvβ3,Bioconjugate Chemistry,2014年,25(2),,393-405
Banerjee, Sangeeta R.; et al,Synthesis and Evaluation of Technetium-99m- and Rhenium-Labeled Inhibitors of the Prostate-Specific Membrane Antigen (PSMA),Journal of Medicinal Chemistry ,2008年,51(15),,4504-4517
Cleeren, Frederik; Lecina, Joan; Billaud, Emilie M. F.; Ahamed, Muneer; Verbruggen, Alfons; Bormans, Guy M.,New Chelators for Low Temperature Al18F-Labeling of Biomolecules,Bioconjugate Chemistry,2016年,27(3),,790-798
Banerjee, Sangeeta Ray; et al,Synthesis and Evaluation of GdIII-Based Magnetic Resonance Contrast Agents for Molecular Imaging of Prostate-Specific Membrane Antigen,Angewandte Chemie, International Edition,2015年,54(37),,10778-10782
Schaefer, Martin; Bauder-Wuest, Ulrike; Leotta, Karin; Zoller, Frederic; Mier, Walter; Haberkorn, Uwe; Eisenhut, Michael; Eder, Matthias,A dimerized urea-based inhibitor of the prostate-specific membrane antigen for 68Ga-PET imaging of prostate cancer,EJNMMI Research,2012年,2(1),,23
Attorney, Agent or Firm:
Kenji Sugimura
Mitsutsugu Sugimura
Mutsumi Yamamoto
Mitsutsugu Sugimura
Mutsumi Yamamoto
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