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Title:
ヒドロキシフェノール誘導体、その調製方法、それらを含む医薬組成物、およびその治療的使用
Document Type and Number:
Japanese Patent JP2008526904
Kind Code:
A
Abstract:
Compounds of the formula (I): in which A, R1, R2, X, Y and Z are defined in the description, the processes for the preparation of these compounds, the uses thereof for the treatment of dyslipidaemia, atherosclerosis and diabetes, and the pharmaceutical compositions comprising them.

Inventors:
Adige, Natalie
Vidal, Katerinu
Zeeuw, Jiang-Jak
Yvon, Stefan
Application Number:
JP2007550706A
Publication Date:
July 24, 2008
Filing Date:
December 22, 2005
Export Citation:
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Assignee:
Merck Patent Gesellschaft mit beschraenkter Haftung
International Classes:
C07C323/22; A61K31/192; A61K31/216; A61K31/421; A61K31/5375; A61P3/06; A61P3/10; A61P9/10; C07C27/02; C07C65/40; C07C67/31; C07C69/94; C07C319/14; C07D263/32; C07D295/08
Domestic Patent References:
JP2001501202A2001-01-30
JPH07173143A1995-07-11
JPS527426A1977-01-20
JPS5265240A1977-05-30
JPS518228A1976-01-23
JPS4892357A1973-11-30
JPH0656740A1994-03-01
JP2004500389A2004-01-08
JPS5732288A1982-02-20
JP2004513076A2004-04-30
JP2003513060A2003-04-08
JPH02221291A1990-09-04
JP2005298437A2005-10-27
JP2007502266A2007-02-08
JP2007536290A2007-12-13
JP2007537301A2007-12-20
JP2009516694A2009-04-23
JP2009516695A2009-04-23
Foreign References:
WO1999011255A11999-03-11
DE4142514A11993-06-24
GB1295447A1972-11-08
US3369025A1968-02-13
US3449325A1969-06-10
GB860303A1961-02-01
WO2004089416A22004-10-21
WO2004089470A22004-10-21
WO2003016254A12003-02-27
GB1098111A1968-01-03
WO1995022323A11995-08-24
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Attorney, Agent or Firm:
Akio Miyazaki
Ishibashi Masayuki
Masaaki Ogata