Title:
11β-ヒドロキシステロイドデヒドロゲナーゼ阻害剤
Document Type and Number:
Japanese Patent JP2011513214
Kind Code:
A
Abstract:
There is provided a compound of formula R1—CO—X—Y—Z—R2 wherein X and Z are each optional groups that are, independently, saturated or unsaturated carbon chains having a length of 1 to 3 carbons; Y is SO, S, SO2, CH═CH, CH2CH2 or O; R1 is wherein denotes the point of attachment; R2 is a heteroaryl group comprising an optionally substituted 5 or 6 membered ring, which ring contains only carbon and at least one nitrogen, or contains only carbon, and at least two nitrogens and at least one sulfur; and wherein (i) when R1 is and —CO—X—Y—Z— is CO—CH2—SO, CO—CH2—S, or CO—CH2—SO2, R2 is other than and; (ii) when R1 is and —CO—X—Y—Z— is —CO—CH2—O—, R2 is other than
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Inventors:
Vicker, Nigel
Sue, Chandon
Prado-Casiano, Fabiennes
Potter, Barry Victor Lloyd
Sue, Chandon
Prado-Casiano, Fabiennes
Potter, Barry Victor Lloyd
Application Number:
JP2010547253A
Publication Date:
April 28, 2011
Filing Date:
February 25, 2009
Export Citation:
Assignee:
Sterix limited
International Classes:
C07D213/30; A61K31/41; A61K31/4164; A61K31/4184; A61K31/4196; A61K31/433; A61K31/44; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4425; A61P1/02; A61P1/04; A61P1/16; A61P3/00; A61P3/04; A61P3/10; A61P7/02; A61P7/04; A61P9/00; A61P9/10; A61P9/12; A61P11/00; A61P11/06; A61P13/12; A61P15/00; A61P17/00; A61P17/02; A61P17/06; A61P19/02; A61P19/10; A61P21/00; A61P21/04; A61P25/00; A61P25/06; A61P25/14; A61P25/16; A61P25/28; A61P27/02; A61P27/16; A61P29/00; A61P31/00; A61P31/04; A61P31/18; A61P35/00; A61P35/02; A61P37/00; A61P37/06; A61P37/08; A61P43/00; C07D213/32; C07D213/34; C07D213/61; C07D213/64; C07D213/65; C07D213/70; C07D213/71; C07D213/80; C07D213/82; C07D213/89; C07D233/84; C07D235/28; C07D249/12; C07D257/04; C07D285/12; C07D285/125; C07D285/135; C07D405/04; C07D409/04
Attorney, Agent or Firm:
Hidesaku Yamamoto
Takaaki Yasumura
Natsuki Morishita
Takaaki Yasumura
Natsuki Morishita