【発明の名称】グルタルイミド抗不安及び抗高血圧剤

Japanese Patent JPH0631222

B2

Glutarimide derivatives of the formula which are useful antihypertensive and antianxiety agents wherein R1 and R2 each independently represent hydrogen, a 1 to 4 carbon alkyl, a 1 to 4 carbon alkoxy, halogen, nitro, hydroxy SO3H, SO2NH2, and when R1 and R2 are taken together, form a fused phenyl group at the 1,2- or 3,4-positions, with the proviso that when R1 and R2 are identical they each represent a hydrogen, a 1 to 4 carbon alkyl, a 1 to 4 carbon alkoxy, hydroxy or a halogen group; A and B independently represent an oxo, a thio or an imino group having the formula -N(R6)- wherein the R6 group is hydrogen or a 1 to 4 carbon alkyl group; R3 is a hydrogen, a 1 to 4 carbon alkyl or hydroxyethyl group; n is an integer of from 2 to 5; and R4 and R5 represent methyl groups or when taken together form a cyclopentane or cyclohexane ring; its enantiomers; and the pharmaceutically acceptable acid addition salts thereof.

MARUSERU HAIBERUTO
MAURISU DABURYUU GITOSU

JP16605985A

April 27, 1994

July 29, 1985

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MERRELL DOW PHARMA

A61K31/435; A61K31/4427; A61K31/443; A61K31/4433; A61K31/445; A61K31/4465; A61K31/45; A61K31/495; A61K31/535; A61K31/54; C07D407/00; A61P9/12; A61P25/20; A61P43/00; C07D221/20; C07D319/00; C07D319/18; C07D401/12; C07D405/12; C07D409/12; C07D411/12; C07D413/12; C07D417/12; (IPC1-7): C07D401/12; A61K31/45; A61K31/495; A61K31/535; A61K31/54; C07D405/12; C07D409/12; C07D411/12; C07D413/12; C07D417/12

Katsuro Sasai

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