Title:
【発明の名称】キノリン-含有α-ケトアミドシステインおよびセリンプロテアーゼインヒビター
Document Type and Number:
Japanese Patent JP2001518506
Kind Code:
A
Abstract:
The present invention is directed to quinoline-containing alpha -ketoamide inhibitors of cysteine and serine proteases are disclosed. Methods for making these compounds, and methods for using the same are also disclosed.
Inventors:
Cheaterj, thunker
Malamo, Jiyoung Pee
Dan, Derek Douglas
J. Joseph, Kurt Allen
Gu, Ji-Kiang
Robert A. Danes
William Dennis, Kingsbury
Pendak, Israel
Siam, Kelvin Sea
Malamo, Jiyoung Pee
Dan, Derek Douglas
J. Joseph, Kurt Allen
Gu, Ji-Kiang
Robert A. Danes
William Dennis, Kingsbury
Pendak, Israel
Siam, Kelvin Sea
Application Number:
JP2000514646A
Publication Date:
October 16, 2001
Filing Date:
October 07, 1998
Export Citation:
Assignee:
Cefalon Incorporated
SmithKline Beach Yam Corporation
SmithKline Beach Yam Corporation
International Classes:
A61K31/47; A61K31/4709; A61K31/517; A61K31/5377; A61K31/55; A61P1/18; A61P7/02; A61P9/10; A61P9/12; A61P11/06; A61P19/02; A61P21/04; A61P25/28; A61P29/00; A61P35/04; A61P43/00; C07D215/40; C07D215/50; C07D239/74; C07D401/12; C07D405/12; C07D409/12; C07D409/14; C07D413/12; C07D417/12; (IPC1-7): C07D215/50; A61K31/47; A61K31/4709; A61K31/517; A61K31/5377; A61K31/55; A61P1/18; A61P7/02; A61P9/10; A61P9/12; A61P11/06; A61P19/02; A61P21/04; A61P25/28; A61P29/00; A61P35/04; A61P43/00; C07D401/12; C07D405/12; C07D409/12; C07D409/14; C07D413/12; C07D417/12
Domestic Patent References:
| JP2001515509A | 2001-09-18 | |||
| JPH08208462A | 1996-08-13 | |||
| JP2001515509A | 2001-09-18 | |||
| JPH08208462A | 1996-08-13 |
Foreign References:
| US5514694A | 1996-05-07 | |||
| US5514694A | 1996-05-07 |
Attorney, Agent or Firm:
Heiyoshi Odashima