【発明の名称】5員複素環縮合ベンゾ誘導体、その調製及び医薬品としてのそれらの使用 - Boehringer Ingelheim Pharma Comandito Gezelshaft

Title:

【発明の名称】5員複素環縮合ベンゾ誘導体、その調製及び医薬品としてのそれらの使用

Document Type and Number:

Japanese Patent JP2002502844

Kind Code:

A

Abstract:

The invention relates to new five-membered, heterocyclic condensed benzoderivatives of the general formula (I), in which Ra to Rc, A, Ar, X and Y have the meanings assigned in claim 1, and their tautomers, stereoisomers, mixtures and salts, especially their physiologically compatible salts with inorganic or organic acids or bases, which have valuable properties. The compounds of the general formula (I) above, in which Rc is a cyano group, present valuable intermediate products for the production of the remaining compounds of the general formula (I), and the compounds of the above general formula (I), in which Rc is one of the following amidino groups, as well as their tautomers and stereoisomers, have valuable pharmacological properties, especially an antithrombotic activity.

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Inventors:

Lies Uwe
Howell norbert
Meme Gerhard
Prepke Henning
Bindel Claus
Stasen Jean Marie
Wienen Wolfgang
Zimmermann Reinell

Application Number:

JP2000530502A

Publication Date:

January 29, 2002

Filing Date:

January 28, 1999

Export Citation:

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Assignee:

Boehringer Ingelheim Pharma Comandito Gezelshaft

International Classes:

C07D277/66; A61K31/403; A61K31/404; A61K31/415; A61K31/4164; A61K31/4184; A61K31/423; A61K31/428; A61K31/4427; A61K31/443; A61K31/4439; A61K31/454; A61K31/4709; A61K31/4725; A61K31/496; A61K31/502; A61K31/5355; A61K31/5377; A61P7/02; A61P9/10; C07D209/14; C07D209/24; C07D235/16; C07D263/56; C07D277/28; C07D277/64; C07D307/81; C07D401/04; C07D401/06; C07D401/08; C07D401/12; C07D401/14; C07D403/04; C07D403/06; C07D403/08; C07D403/12; C07D403/14; C07D405/12; C07D405/14; C07D417/12; C07F9/32; C07F9/6506; (IPC1-7): C07D235/16; A61K31/403; A61K31/404; A61K31/415; A61K31/4164; A61K31/4184; A61K31/423; A61K31/428; A61K31/4439; A61K31/454; A61K31/4709; A61K31/4725; A61K31/496; A61K31/502; A61K31/5377; A61P7/02; A61P9/10; C07D209/14; C07D263/56; C07D277/66; C07D307/81; C07D401/04; C07D401/12; C07D401/14; C07D403/04; C07D403/06; C07D403/08; C07D403/12; C07D403/14; C07D405/12; C07D405/14; C07D417/12; C07F9/32

Attorney, Agent or Firm:

Minoru Nakamura (9 outside)

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