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Title:
抗コリン作用薬を含有する吸入用エアロゾル製剤
Document Type and Number:
Japanese Patent JP4602767
Kind Code:
B2
Abstract:
Aqueous composition (A) for inhalation contains as only active ingredient a tricyclo-oxa-aza-nonane derivative (I), at least one acid and optionally other auxiliaries and/or complexing agents. Aqueous composition (A) for inhalation contains as only active ingredient a tricylo-oxa-aza-nonane derivative of formula (I), at least one acid and optionally other auxiliaries and/or complexing agents. [Image] X : chloride, bromide, iodide, sulfate, phosphate, methanesulfonate, nitrate, maleate, acetate, citrate, fumarate, tartrate, oxalate, succinate, benzoate or p-toluenesulfonate. An independent claim is also included for an inhalation kit containing (A) and an inhaler for nebulization. ACTIVITY : Antiasthmatic. No details of tests for antiasthmatic activity are given. MECHANISM OF ACTION : Anticholinergic.

Inventors:
Schmid friedrich
Application Number:
JP2004533274A
Publication Date:
December 22, 2010
Filing Date:
July 25, 2003
Export Citation:
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Assignee:
Boehringer Ingelheim Pharma Gesellshaft Mitt Beschlenktel Haftung Und Company Comandito Gesellshaft
International Classes:
A61K31/46; A61K9/00; A61K9/12; A61K9/72; A61K31/33; A61K31/5375; A61K47/04; A61K47/12; A61K47/18; A61K47/22; A61M15/00; A61P11/00; A61P11/06; A61P43/00
Domestic Patent References:
JP5509241A
JP11512649A
Foreign References:
WO2002032899A1
WO2002049624A1
Attorney, Agent or Firm:
Sadao Kumakura
Nobuo Ogawa
Atsushi Hakoda
Kenji Asai
Koji Hirayama