Title:
INHIBITOR OF HISTONE DEACETYLASE
Document Type and Number:
Japanese Patent JP2005255683
Kind Code:
A
Abstract:
To provide a composition having activities for inhibiting a histone deacetylase, and usable for treating cell proliferation disease.
For example, a compound having formula (I) (wherein, J is a 1-3C hydrocarbon chain, -NHCH2- or the like; and X and Y are each an amino group, a substituted amino group, a heterocycle containing N, or the like) or formula (II) (wherein, Ar3 is an arylene or a heteroarylene; X is an alkylene, -CH2-NH-, -CH2-S- or the like; and Cy3 is an aryl, a heteroaryl or the like) has the above activities.
Inventors:
DELORME DANIEL
WOO SOON HYUNG
VAISBURG ARKADII
MORADEI OSCAR
LEIT SILVANA
RAEPPEL STEPHANE
FRECHETTE SYLVIE
BOUCHAIN GILIANE
WOO SOON HYUNG
VAISBURG ARKADII
MORADEI OSCAR
LEIT SILVANA
RAEPPEL STEPHANE
FRECHETTE SYLVIE
BOUCHAIN GILIANE
Application Number:
JP2005080310A
Publication Date:
September 22, 2005
Filing Date:
March 18, 2005
Export Citation:
Assignee:
METHYLGENE INC
International Classes:
C07D251/46; A61K31/167; A61K31/17; A61K31/18; A61K31/277; A61K31/34; A61K31/343; A61K31/352; A61K31/357; A61K31/36; A61K31/381; A61K31/4035; A61K31/4045; A61K31/407; A61K31/41; A61K31/415; A61K31/4164; A61K31/4184; A61K31/421; A61K31/423; A61K31/4245; A61K31/426; A61K31/428; A61K31/437; A61K31/44; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4418; A61K31/4436; A61K31/4439; A61K31/444; A61K31/454; A61K31/455; A61K31/47; A61K31/4709; A61K31/472; A61K31/495; A61K31/496; A61P35/00; A61P43/00; C07C233/44; C07C233/80; C07C235/38; C07C235/42; C07C235/56; C07C235/82; C07C235/84; C07C237/20; C07C237/22; C07C237/40; C07C237/42; C07C255/58; C07C255/59; C07C275/34; C07C275/36; C07C311/42; C07C323/32; C07C323/36; C07C323/44; C07C323/60; C07C381/00; C07D209/14; C07D209/46; C07D211/88; C07D213/30; C07D213/38; C07D213/44; C07D213/56; C07D213/70; C07D213/74; C07D213/75; C07D213/81; C07D213/82; C07D213/85; C07D215/22; C07D215/36; C07D215/38; C07D215/48; C07D217/04; C07D231/12; C07D231/38; C07D233/54; C07D233/64; C07D233/84; C07D235/26; C07D235/28; C07D235/30; C07D239/36; C07D239/42; C07D239/47; C07D239/52; C07D239/91; C07D239/96; C07D251/18; C07D251/48; C07D251/50; C07D251/52; C07D251/54; C07D251/70; C07D251/72; C07D253/08; C07D257/04; C07D263/14; C07D263/22; C07D263/24; C07D263/58; C07D265/26; C07D265/36; C07D271/06; C07D271/10; C07D277/20; C07D277/30; C07D277/42; C07D277/70; C07D277/74; C07D277/82; C07D279/16; C07D295/12; C07D295/14; C07D295/155; C07D307/12; C07D307/16; C07D307/28; C07D307/85; C07D311/04; C07D311/22; C07D311/56; C07D311/58; C07D311/74; C07D317/66; C07D319/18; C07D319/20; C07D333/20; C07D333/36; C07D333/38; C07D333/70; C07D401/04; C07D401/12; C07D403/04; C07D405/12; C07D409/12; C07D413/12; C07D417/12; C07D473/16; C07D473/34; C07D473/40; C07D487/04; C07D491/113; C07D495/04; C07D498/04; C07D513/04; C07D521/00; C07F7/08; C07F7/10; C07F7/18; C12N9/99; (IPC1-7): C07D251/70; A61K31/167; A61K31/18; A61K31/277; A61K31/34; A61K31/343; A61K31/36; A61K31/381; A61K31/4035; A61K31/4045; A61K31/407; A61K31/41; A61K31/415; A61K31/421; A61K31/423; A61K31/4245; A61K31/426; A61K31/428; A61K31/44; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4418; A61K31/4436; A61K31/4439; A61K31/444; A61K31/45; A61K31/454; A61K31/455; A61K31/47; A61K31/4745; A61K31/495; A61K31/496; A61K31/505; A61K31/506; A61K31/517; A61K31/519; A61K31/52; A61K31/53; A61K31/536; A61K31/5375; A61K31/5377; A61K31/538; A61K31/5383; A61K31/5415; A61K31/695; A61P35/00; A61P43/00; C07C233/11; C07C233/80; C07C235/38; C07C235/42; C07C235/56; C07C235/82; C07C235/84; C07C237/20; C07C237/22; C07C237/32; C07C237/42; C07C255/58; C07C255/59; C07C271/28; C07C275/36; C07C311/39; C07C323/36; C07C323/44; C07C323/60; C07D209/14; C07D209/46; C07D209/48; C07D211/88; C07D213/30; C07D213/36; C07D213/56; C07D213/70; C07D213/74; C07D213/75; C07D213/81; C07D213/82; C07D213/85; C07D215/36; C07D215/38; C07D215/48; C07D217/04; C07D231/12; C07D231/38; C07D233/84; C07D239/36; C07D239/38; C07D239/42; C07D239/52; C07D239/88; C07D239/91; C07D239/96; C07D251/46; C07D251/48; C07D251/50; C07D251/52; C07D251/72; C07D253/08; C07D257/04; C07D263/14; C07D263/22; C07D263/58; C07D265/26; C07D265/36; C07D271/06; C07D271/10; C07D277/20; C07D277/42; C07D277/68; C07D277/74; C07D277/82; C07D279/16; C07D295/12; C07D307/16; C07D307/28; C07D307/85; C07D311/74; C07D317/66; C07D319/18; C07D319/20; C07D333/20; C07D333/36; C07D333/38; C07D401/04; C07D401/12; C07D403/04; C07D405/12; C07D409/12; C07D413/12; C07D417/12; C07D473/16; C07D473/40; C07D487/04; C07D491/113; C07D495/04; C07D498/04; C07F7/18; C12N9/99
Domestic Patent References:
JPH10152462A | 1998-06-09 | |||
JPH11269146A | 1999-10-05 | |||
JP3795044B2 | 2006-07-12 |
Foreign References:
WO2001038322A1 | 2001-05-31 | |||
WO2001016106A1 | 2001-03-08 |
Attorney, Agent or Firm:
Hideto Asamura
Hajime Asamura
Naganuma Akio
Yukihiro Ikeda
Hajime Asamura
Naganuma Akio
Yukihiro Ikeda