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Title:
インスリン受容体部分アゴニスト
Document Type and Number:
Japanese Patent JP2018501203
Kind Code:
A
Abstract:
インスリン受容体において部分アゴニストとして作用するインスリン二量体およびインスリンアナログ二量体が開示される。【選択図】図1

Inventors:
Lynn, Sonnien
Yang, Lin
Fo, pay
Pisarnicki, Dmitry
Fen, tantin
Navy, Ravi
Ju, Yupin
Kecketts, Ahmed
Madsen-Dugan, Christina Bee
See, Gee-Tsai
Woo, Zee Tsai
Mu, Einjuin
Application Number:
JP2017526961A
Publication Date:
January 18, 2018
Filing Date:
November 19, 2015
Export Citation:
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Assignee:
Merck Sharp & Dohme Corp.
International Classes:
C07K19/00; A61K38/28; A61K47/54; A61K47/60; A61P3/10; C07K14/62
Foreign References:
WO2014052451A22014-04-03
WO2008145721A22008-12-04
Other References:
NAUNYN-SCHMIEDEBERG'S ARCHIVES OF PHARMACOLOGY, vol. VOL:350, NR:2, JPN5017009928, August 1994 (1994-08-01), pages PAGE(S):213 - 217
HOPPE-SEYLER'S ZEITSCHRIFT FUER PHYSIOLOGISCHE CHEMIE, vol. VOL:363, NR:3, JPN5017009929, March 1982 (1982-03-01), pages PAGE(S):317 - 330
BIOCHEMICAL PHARMACOLOGY, 1989年, vol. 38, no. 14, JPN6018024313, pages 2269 - 2277
DIABETOLOGIA, 1995年, vol. Vol.38, JPN6018024314, pages 1007 - 1013
Attorney, Agent or Firm:
Makoto Ono
Kenkyo Kanayama
Mitsuaki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Takahiro Aoki
Yoshie Sakurada
Yousuke Kawasaki
Takuya Gomibuchi
Toshikazu Imato
Yoichi Iino
Yusuke Ichikawa
Masahiro Moriyama
Yoshikazu Iwase
Yasufumi Shiroyama