Title:
好中球依存性炎症性疾患の治療におけるキラルアリールケトン
Document Type and Number:
Japanese Patent JP5021169
Kind Code:
B2
Abstract:
The compounds of formula (I): where Ar is an aromatic ring and Ra, Rb, are as defined in the description, are useful in therapy as drugs for the treatment of diseases mediated by infiltrations of neutrophils induced by IL-8, such as psoriasis, rheumatoid arthritis, ulcerative cholitis and for the treatment of damages caused by ischemia and reperfusion.
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Inventors:
Alegretti, Marcello
Bertini, ricardo
Chester, Maria Candida
Bizari, chinsia
Colotta, Francesco
Bertini, ricardo
Chester, Maria Candida
Bizari, chinsia
Colotta, Francesco
Application Number:
JP2004558041A
Publication Date:
September 05, 2012
Filing Date:
December 09, 2003
Export Citation:
Assignee:
Dompe Fa.le.Ma Sochieta per Azioni
International Classes:
A61K31/12; A61K31/19; A61K31/215; A61K31/222; A61P1/04; A61P9/10; A61P11/00; A61P13/12; A61P17/00; A61P17/06; A61P29/00; A61P43/00; C07C45/56; C07C45/67; C07C49/213; C07C49/215; C07C49/782; C07C49/784; C07C69/612; C07C69/738; C07C69/78; C07C271/18; C07C309/65; C07C311/21; C07C317/06; C07C317/24; C07D209/46; C07D213/50; C07D319/06; C07F9/40; C07C65/32
Domestic Patent References:
JP2003522750A | ||||
JP2002528434A |
Other References:
G.Picciola, et al.,FARMACO ED. SCI.,1981年,Vol.36, No. 12,p.1037-1056
Attorney, Agent or Firm:
Shinjiro Ono
Kazuo Shamoto
Tadashi Masui
Yasushi Kobayashi
Akio Chiba
Hiroyuki Tomita
Kazuo Shamoto
Tadashi Masui
Yasushi Kobayashi
Akio Chiba
Hiroyuki Tomita