Title:
オレキシン受容体拮抗薬として有用なラクタム誘導体
Document Type and Number:
Japanese Patent JP5847830
Kind Code:
B2
Abstract:
The present invention relates to lactam derivatives of formula (I) wherein Y, R1, R2 and R3 are as described in the description, to their preparation, to pharmaceutically acceptable salts thereof, and to their use as pharmaceuticals, to pharmaceutical compositions containing one or more compounds of formula (I), and especially to their use as orexin receptor antagonists.
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Inventors:
Hamed Aisa Oui
Christoph Boss
Christine blotch
Bivia Hydeman
Thierry Schifferlen
Jody Tea Williams
Christoph Boss
Christine blotch
Bivia Hydeman
Thierry Schifferlen
Jody Tea Williams
Application Number:
JP2013538312A
Publication Date:
January 27, 2016
Filing Date:
November 09, 2011
Export Citation:
Assignee:
Actelion Pharmaceuticals Ltd
International Classes:
C07D207/26; A61K31/4015; A61K31/4025; A61K31/403; A61K31/404; A61K31/4155; A61K31/4192; A61K31/4245; A61K31/427; A61K31/428; A61K31/4439; A61K31/45; A61K31/4525; A61K31/4535; A61K31/454; A61K31/4545; A61K31/4709; A61K31/495; A61K31/498; A61K31/506; A61K31/5375; A61K31/5377; A61K31/55; A61P25/20; A61P25/28; A61P25/30; A61P43/00; C07D211/76; C07D223/10; C07D241/08; C07D265/32; C07D401/06; C07D401/10; C07D401/14; C07D403/06; C07D403/10; C07D405/06; C07D405/14; C07D409/06; C07D413/04; C07D413/06; C07D413/10; C07D413/14; C07D417/06; C07D417/10; C07D417/14; C07D471/04
Domestic Patent References:
| JP2005501026A | ||||
| JP2006501201A |
Foreign References:
| WO2010048014A1 |
Attorney, Agent or Firm:
Mitsue Obuchi
Yukio Fuse
Yukio Fuse