MANUFACTURING METHOD OF 1,2,4-OXADIAZOLE DERIVATIVE

Title:

MANUFACTURING METHOD OF 1,2,4-OXADIAZOLE DERIVATIVE

Document Type and Number:

Japanese Patent JP2007084449

Kind Code:

A

Abstract:

To provide a method for manufacturing an aimed 1,2,4-oxadiazole derivative from an O-acylamidoxime compound bearing an easily hydrolyzable substituent group in a high yield by simple purification while suppressing side reactions.

The manufacturing method of the 1,2,4-oxadiazole derivative represented by general formula (II) comprises subjecting the O-acylamidoxime compound represented by general formula (I) [wherein R1 and R2 are each independently a substituted or unsubstituted alkyl, alkenyl, alkynyl, aryl or heterocyclic group] to a ring closure reaction in the presence of a cyclic acid anhydride.

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Inventors:

TAKAHASHI MAKOTO

Application Number:

JP2005271999A

Publication Date:

April 05, 2007

Filing Date:

September 20, 2005

Export Citation:

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Assignee:

FUJIFILM CORP

International Classes:

C07D271/06

Attorney, Agent or Firm:

Shohei Oguri
Hironori Honda
Toshimitsu Ichikawa
Takeshi Takamatsu
Kiyozumi Yazawa

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