Title:
4-(ビフェニリル)アゼチジン-2-オンホスホン酸類の製造方法
Document Type and Number:
Japanese Patent JP2008545700
Kind Code:
A
Abstract:
The present invention relates to processes for the production of 4-(biphenylyl)azetidin-2-one phosphonic acid derivatives of formula
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Inventors:
Antonelli Stefan
Baden Timothy C.
Lee Peter
Martinez Eduard
SCHAIRER WAYNE C.
TALLEY JOHN J.
Baden Timothy C.
Lee Peter
Martinez Eduard
SCHAIRER WAYNE C.
TALLEY JOHN J.
Application Number:
JP2008513703A
Publication Date:
December 18, 2008
Filing Date:
May 25, 2006
Export Citation:
Assignee:
MICROBIA, INC.
International Classes:
C07D205/08; C07D263/26; C07F5/02; C07F7/18; C07F9/568; C07F9/6596; C07F19/00; C07B61/00
Domestic Patent References:
| JPH06508637A | 1994-09-29 | |||
| JP2005053931A | 2005-03-03 | |||
| JP2004516280A | 2004-06-03 | |||
| JP2008542205A | 2008-11-27 | |||
| JP2008540557A | 2008-11-20 |
Foreign References:
| WO2002066464A1 | 2002-08-29 |
Other References:
JPN6012022029; ＣＬＡＤＥＲ，Ｊ．Ｗ． ｅｔ ａｌ: '２-Ａｚｅｔｉｄｉｎｏｎｅ Ｃｈｏｌｅｓｔｅｒｏｌ Ａｂｓｏｒｐｔｉｏｎ Ｉｎｈｉｂｉｔｏｒｓ： Ｓｔｒｕｃｔｕｒｅ-Ａｃｔｉｖｉｔｙ Ｒｅｌａｔｉｏｎｓｈｉｐｓ ｏｎ ｔｈｅ Ｈｅｔｅｒｏｃｙｃｌｉ' Ｊｏｕｒｎａｌ ｏｆ Ｍｅｄｉｃｉｎａｌ Ｃｈｅｍｉｓｔｒｙ Ｖｏｌ．３９， Ｎｏ．１９, 1996, ｐ．３６８４-３６９３
JPN6012022032; ＶＡＣＣＡＲＯ，Ｗ．Ｄ． ｅｔ ａｌ: '２-ａｚｅｔｉｄｉｎｏｎｅ ｃｈｏｌｅｓｔｅｒｏｌ ａｂｓｏｒｐｔｉｏｎ ｉｎｈｉｂｉｔｏｒｓ： ｉｎｃｒｅａｓｅｄ ｐｏｔｅｎｃｙ ｂｙ ｓｕｂｓｔｉｔｕｔｉｏｎ ｏｆ ｔｈｅ Ｃ-４ ｐｈｅｎｙｌ' Ｂｉｏｏｒｇａｎｉｃ ＆ Ｍｅｄｉｃｉｎａｌ Ｃｈｅｍｉｓｔｒｙ Ｖｏｌ．６， Ｎｏ．９, 1998, ｐ．１４２９-１４３７
JPN6012022032; ＶＡＣＣＡＲＯ，Ｗ．Ｄ． ｅｔ ａｌ: '２-ａｚｅｔｉｄｉｎｏｎｅ ｃｈｏｌｅｓｔｅｒｏｌ ａｂｓｏｒｐｔｉｏｎ ｉｎｈｉｂｉｔｏｒｓ： ｉｎｃｒｅａｓｅｄ ｐｏｔｅｎｃｙ ｂｙ ｓｕｂｓｔｉｔｕｔｉｏｎ ｏｆ ｔｈｅ Ｃ-４ ｐｈｅｎｙｌ' Ｂｉｏｏｒｇａｎｉｃ ＆ Ｍｅｄｉｃｉｎａｌ Ｃｈｅｍｉｓｔｒｙ Ｖｏｌ．６， Ｎｏ．９, 1998, ｐ．１４２９-１４３７
Attorney, Agent or Firm:
Kenichi Morita
Kenjiro Yamaguchi
Kenjiro Yamaguchi