Title:
三環式化合物の製造方法
Document Type and Number:
Japanese Patent JP2021527691
Kind Code:
A
Abstract:
本発明は、X、R1、R2、R3、R4、U、A1、A2、A3およびA4が上記のように定義される式(II)の化合物から出発して式(I)の化合物を調製する方法に関する。本発明はさらに、式(III)および(IV)の化合物(ここで、全ての変数は、上記で定義された通りである)に関する。【化1】
Inventors:
Lenbiark, Andreas
Hail, Keira
Steiff, Andreas Karl
Ford, Marc James
Hail, Keira
Steiff, Andreas Karl
Ford, Marc James
Application Number:
JP2020570919A
Publication Date:
October 14, 2021
Filing Date:
June 17, 2019
Export Citation:
Assignee:
Bayer Actien Gezershyaft
International Classes:
C07D401/04; C07F1/02; C07F3/02; C07F3/06
Foreign References:
WO2016174052A1 | 2016-11-03 |
Other References:
HUANG, ZHIHONG ET AL.: "Palladium-Catalyzed Cross-Coupling Reactions with Zinc, Boron, and IndiumExhibiting High Turnover Nu", ORGANOMETALLICS, vol. 24, no. 4, JPN6023021659, 2005, pages 475 - 478, XP001236762, ISSN: 0005227398, DOI: 10.1021/om049106j
XU, SHIQING ET AL.: "Pd-catalyzedcross-coupling reactions exhibiting catalyst turnover numbers(TONs) exceedingone million", ARKIVOC, JPN6023021660, 2012, pages 242 - 252, ISSN: 0005227399
YANG, YANG ET AL.: "Mild and generalconditions for Negishi cross-coupling enabled by the use of palladacycleprecatalysts", ANGEWANDTE CHEMIE, INTERNATIONAL EDITION, vol. 52, no. 2, JPN6023021661, 2013, pages 615 - 619, ISSN: 0005227400
XU, SHIQING ET AL.: "Pd-catalyzedcross-coupling reactions exhibiting catalyst turnover numbers(TONs) exceedingone million", ARKIVOC, JPN6023021660, 2012, pages 242 - 252, ISSN: 0005227399
YANG, YANG ET AL.: "Mild and generalconditions for Negishi cross-coupling enabled by the use of palladacycleprecatalysts", ANGEWANDTE CHEMIE, INTERNATIONAL EDITION, vol. 52, no. 2, JPN6023021661, 2013, pages 615 - 619, ISSN: 0005227400
Attorney, Agent or Firm:
Makoto Ono
Kenkyo Kanayama
Mitsuaki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Yoshie Sakurada
Yousuke Kawasaki
Takuya Gomibuchi
Yoichi Iino
Yusuke Ichikawa
Masahiro Moriyama
Takashi Kono
Yoshikazu Iwase
Yasufumi Shiroyama
Kenkyo Kanayama
Mitsuaki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Yoshie Sakurada
Yousuke Kawasaki
Takuya Gomibuchi
Yoichi Iino
Yusuke Ichikawa
Masahiro Moriyama
Takashi Kono
Yoshikazu Iwase
Yasufumi Shiroyama