Title:
METHODS, COMPOUNDS, COMPOSITIONS AND VEHICLES FOR DELIVERING 3-AMINO-1-PROPANESULFONIC ACID
Document Type and Number:
Japanese Patent JP2016222671
Kind Code:
A
Abstract:
PROBLEM TO BE SOLVED: To provide methods, compounds, compositions and vehicles for delivering 3-amino-1-propanesulfonic acid (3APS) in a human subject, and to provide compounds that yield or generate 3APS, either in vitro or in vivo.SOLUTION: This invention relates to a compound expressed by e.g. formula I-A, and a pharmaceutically acceptable salt. (Rx and Ry are each independently selected from H and a protecting group; Rx and Ry are not both H at the same time; and L1 and L2 are each a cleavable linkage; and when Rx is H, L1 is absent, and when Ry is H, then L2 is absent).SELECTED DRAWING: None
Inventors:
KONG XIANQI
MOHAMED ATFANI
BENOIT BACHAND
ABDERRAHIM BOUZIDE
STEPHANE CIBLAT
SOPHIE LEVESQUE
DAVID MIGNEAULT
ISABELLE VALADE
WU XINFU
DANIEL DELORME
MOHAMED ATFANI
BENOIT BACHAND
ABDERRAHIM BOUZIDE
STEPHANE CIBLAT
SOPHIE LEVESQUE
DAVID MIGNEAULT
ISABELLE VALADE
WU XINFU
DANIEL DELORME
Application Number:
JP2016111832A
Publication Date:
December 28, 2016
Filing Date:
June 03, 2016
Export Citation:
Assignee:
BHI LP
International Classes:
C07C309/15; A61P25/28; C07C401/00; C07D207/16; C07D209/20; C07D217/24; C07D233/64; C07D307/62; C07D317/40; C07D333/24; C07H5/04; C07H13/12; C07H15/04; C07J41/00
Domestic Patent References:
| JPS6242998A | 1987-02-24 |
Foreign References:
| WO2004113275A2 | 2004-12-29 | |||
| WO2006085149A2 | 2006-08-17 | |||
| WO2004113391A2 | 2004-12-29 | |||
| WO2004058258A1 | 2004-07-15 | |||
| WO2004058239A1 | 2004-07-15 |
Attorney, Agent or Firm:
Ryoichi Takaoka