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Patent Searching and Data


Title:
方法および中間体
Document Type and Number:
Japanese Patent JP2013528624
Kind Code:
A
Abstract:
A process for preparing enantioselectively a compound of formula I-1a or I-1b: over a compound of formulas I-2-I-7:

Inventors:
Gerald Jay Tanoury
Application Number:
JP2013513371A
Publication Date:
July 11, 2013
Filing Date:
June 03, 2011
Export Citation:
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Assignee:
VERTEX PHARMACEUTICALS INCORPORATED
International Classes:
C07D209/52; C07D471/18; C12P21/02; C07K5/107
Domestic Patent References:
JP2009504780A2009-02-05
JPS6013756A1985-01-24
Other References:
JPN6015011791; Organic Letters 7(20), 2005, 4337-4340
JPN6015011794; Tetrahedron Letters 49, 2008, 6327-6329
JPN6015011797; J.Am.Chem.Soc. 132(21), 2010, 7260-7261
JPN6015011799; Organic Letters 11(9), 2009, 1935-1938
JPN6015011802; Tetrahedron Letters 47, 2006, 6469-6472
Attorney, Agent or Firm:
Aoyama Aoi
Takuji Yamada
Michiko Matsutani
Mitsutaka Iwasaki
Yasushi Ochiai