Title:
血漿カリクレイン阻害剤としてのN−((6−アミノ−ピリジン−3−イル)メチル)−ヘテロアリール−カルボキサミド類
Document Type and Number:
Japanese Patent JP5809267
Kind Code:
B2
Abstract:
The invention relates to compound of the formula I in which the substituents are as defined in the specification; in free form or in salt form; to its preparation, to its use as medicament and to medicaments comprising it.
Inventors:
Trixie Brandle
Stephanie Flore
Sebastian Kopek
Julie Lachar
Christian Markert
Kenji Namoto
Perluru Nangaga
Bernard Pilar
Martin Lenatus
Richard Cedrani
Thomas Tooler
Stephanie Flore
Sebastian Kopek
Julie Lachar
Christian Markert
Kenji Namoto
Perluru Nangaga
Bernard Pilar
Martin Lenatus
Richard Cedrani
Thomas Tooler
Application Number:
JP2013522243A
Publication Date:
November 10, 2015
Filing Date:
August 03, 2011
Export Citation:
Assignee:
Novartis Age
International Classes:
C07D401/12; A61K31/443; A61K31/4439; A61K31/444; A61K31/4545; A61K31/4709; A61K31/4725; A61K31/497; A61K31/498; A61K31/506; A61K31/5377; A61K31/538; A61K45/00; A61P3/10; A61P7/10; A61P9/10; A61P9/12; A61P43/00; C07D401/14; C07D405/12; C07D405/14; C07D409/14; C07D413/12; C07D413/14; C07D417/12; C07D417/14; C07D471/04; C07D495/04
Domestic Patent References:
JP2009545611A | ||||
JP2005517734A | ||||
JP2004509067A |
Foreign References:
WO2001079261A1 |
Attorney, Agent or Firm:
Hiroshi Kobayashi
Norio Omori
Yasuhito Suzuki
Norio Omori
Yasuhito Suzuki