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Title:
血漿カリクレイン阻害剤としてのN−((6−アミノ−ピリジン−3−イル)メチル)−ヘテロアリール−カルボキサミド類
Document Type and Number:
Japanese Patent JP5809267
Kind Code:
B2
Abstract:
The invention relates to compound of the formula I in which the substituents are as defined in the specification; in free form or in salt form; to its preparation, to its use as medicament and to medicaments comprising it.

Inventors:
Trixie Brandle
Stephanie Flore
Sebastian Kopek
Julie Lachar
Christian Markert
Kenji Namoto
Perluru Nangaga
Bernard Pilar
Martin Lenatus
Richard Cedrani
Thomas Tooler
Application Number:
JP2013522243A
Publication Date:
November 10, 2015
Filing Date:
August 03, 2011
Export Citation:
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Assignee:
Novartis Age
International Classes:
C07D401/12; A61K31/443; A61K31/4439; A61K31/444; A61K31/4545; A61K31/4709; A61K31/4725; A61K31/497; A61K31/498; A61K31/506; A61K31/5377; A61K31/538; A61K45/00; A61P3/10; A61P7/10; A61P9/10; A61P9/12; A61P43/00; C07D401/14; C07D405/12; C07D405/14; C07D409/14; C07D413/12; C07D413/14; C07D417/12; C07D417/14; C07D471/04; C07D495/04
Domestic Patent References:
JP2009545611A
JP2005517734A
JP2004509067A
Foreign References:
WO2001079261A1
Attorney, Agent or Firm:
Hiroshi Kobayashi
Norio Omori
Yasuhito Suzuki