Title:
新しい抗菌性化合物
Document Type and Number:
Japanese Patent JP2019517546
Kind Code:
A
Abstract:
本発明は、新規な抗菌化合物、それらを含有する医薬組成物、および抗菌剤としてのそれらの使用に関する。
Inventors:
Ombrat Rocera
Magaro Gabriele
Garofalo Barbara
Furlotti Guido
Mangano Giorgina
Capezone de joanon alessandra
Magaro Gabriele
Garofalo Barbara
Furlotti Guido
Mangano Giorgina
Capezone de joanon alessandra
Application Number:
JP2018564240A
Publication Date:
June 24, 2019
Filing Date:
June 05, 2017
Export Citation:
Assignee:
AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F.SOCIETA PER AZIONI
International Classes:
C07D401/14; A61K31/4375; A61K31/4545; A61K31/4709; A61K31/4725; A61K31/498; A61K31/4985; A61K31/536; A61K31/5377; A61K31/5383; A61K31/542; A61P31/04; C07D471/04; C07D491/052; C07D498/04; C07D519/00
Domestic Patent References:
JPH05170743A | 1993-07-09 | |||
JP2009149618A | 2009-07-09 | |||
JP2011520943A | 2011-07-21 | |||
JP2011520944A | 2011-07-21 | |||
JP2010526130A | 2010-07-29 | |||
JP2008542249A | 2008-11-27 | |||
JP2014518267A | 2014-07-28 | |||
JP6723242B2 | 2020-07-15 | |||
JP2017537938A | 2017-12-21 | |||
JP2019517545A | 2019-06-24 |
Foreign References:
WO2006046552A1 | 2006-05-04 | |||
CN105218501A | 2016-01-06 | |||
WO2016027249A1 | 2016-02-25 |
Other References:
BOBESH, KARYAKULAM ANDREWS; RENUKA, JANUPALLY; SRILAKSHMI, RUDRARAJU RESHMA; YELLANKI, SWAPNA; KULKA: "Replacement of cardiotoxic aminopiperidine linker with piperazine moiety reduces cardiotoxicity? Myc", BIOORGANIC & MEDICINAL CHEMISTRY, vol. 24(1),, JPN6021016919, 2016, pages 42 - 52, ISSN: 0004649547
第5版実験化学講座13, JPN6021016921, 20 February 2004 (2004-02-20), pages 295 - 297, ISSN: 0004649548
BOBESH, KARYAKULAM ANDREWS; RENUKA, JANUPALLY; JEANKUMAR, VARIAM ULLAS; SHRUTI, SINGH KAKAN; SRIDEVI: "Extending the N-linked aminopiperidine class to the mycobacterial gyrase domain: Pharmacophore mappi", EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 85,, JPN6021016923, 2014, pages 593 - 604, ISSN: 0004501953
KAMAL, A.; SATYANARAYANA, M.; DEVAIAH, V.; ROHINI, V.; YADAV, J. S.; MULLICK, B.; NAGARAJA, V.: "Synthesis and biological evaluation of coumarin linked fluoroquinolones, phthalimides and naphthalim", LETTERS IN DRUG DESIGN & DISCOVERY, vol. 3(7),, JPN6021016924, 2006, pages 494 - 502, ISSN: 0004501954
第5版実験化学講座13, JPN6021016921, 20 February 2004 (2004-02-20), pages 295 - 297, ISSN: 0004649548
BOBESH, KARYAKULAM ANDREWS; RENUKA, JANUPALLY; JEANKUMAR, VARIAM ULLAS; SHRUTI, SINGH KAKAN; SRIDEVI: "Extending the N-linked aminopiperidine class to the mycobacterial gyrase domain: Pharmacophore mappi", EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 85,, JPN6021016923, 2014, pages 593 - 604, ISSN: 0004501953
KAMAL, A.; SATYANARAYANA, M.; DEVAIAH, V.; ROHINI, V.; YADAV, J. S.; MULLICK, B.; NAGARAJA, V.: "Synthesis and biological evaluation of coumarin linked fluoroquinolones, phthalimides and naphthalim", LETTERS IN DRUG DESIGN & DISCOVERY, vol. 3(7),, JPN6021016924, 2006, pages 494 - 502, ISSN: 0004501954
Attorney, Agent or Firm:
Patent Service Corporation Patent Office Sykes