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Title:
新規イミダゾ[1,2−a]ピリジン及びイミダゾ[1,2−b]ピリダジン誘導体
Document Type and Number:
Japanese Patent JP5643105
Kind Code:
B2
Abstract:
Imidazo[1,2-a]pyridine and imidazo[1,2-b]pyridazine derivatives which inhibit Btk and are useful for the treatment of auto-immune and inflammatory diseases caused by aberrant B-cell activation, e.g. arthritis.

Inventors:
デュードニー,ノーラン・ジェームス
ロウ,イェン
ソス,マイケル
Application Number:
JP2010537386A
Publication Date:
December 17, 2014
Filing Date:
December 04, 2008
Export Citation:
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Assignee:
エフ.ホフマン−ラ ロシュ アーゲーF. HOFFMANN−LA ROCHE AKTIENGESELLSCHAFT
International Classes:
C07D471/04; A61K31/437; A61K31/444; A61K31/455; A61K31/496; A61K31/5025; A61K31/506; A61K31/5377; A61K31/541; A61K31/55; A61K31/551; A61K31/695; A61P19/02; A61P29/00; A61P37/06; A61P43/00; C07D487/04; C07D519/00; C07F7/10
Attorney, Agent or Firm:
Patent business corporation Tsukuni
Hajime Tsukuni
Ito 佐保子
Toshio Miyake
Akio Shibata
Yasuhiro Kokuni
Yoko Tanaka
Yoshinori Ubukawa