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Title:
窒素含有縮合環化合物及びその用途
Document Type and Number:
Japanese Patent JP3988832
Kind Code:
B2
Abstract:

To provide an excellent URAT1 (urate transporter 1) activity inhibitor effective in treatment, etc., of pathological conditions in which uric acid is associated such as hyperuricemia, gouty node, acute gouty arthritis, chronic gouty arthritis, gouty kidney, urinary calculus, renal dysfunction, coronary artery disease and ischemic heart disease.

The URAT1 activity inhibitor comprises the nitrogen-containing condensed ring compound represented by general formula [1] or its pharmaceutically acceptable salt as an active ingredient.

COPYRIGHT: (C)2006,JPO&NCIPI


Inventors:
Kazuyuki Hirata
Naoki Ogawa
Shinagawa Yukou
Toshihiro Kiguchi
Teruhiko Inoue
Akira Matsuo
Yoshinori Kosugi
Nomura Yukihiro
Koichiro Kawahara
Uehara Hideto
Application Number:
JP2005343214A
Publication Date:
October 10, 2007
Filing Date:
November 29, 2005
Export Citation:
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Assignee:
Japan Tobacco Inc.
International Classes:
C07D265/36; A61K31/538; A61K31/5383; A61P9/00; A61P9/10; A61P13/04; A61P13/12; A61P19/02; A61P19/06; A61P43/00; C07D498/04; A61K31/404; A61K31/47; A61K31/498; A61K31/5415; A61K31/55; A61K31/5513; A61K31/553; C07D209/08; C07D215/08; C07D223/16; C07D241/42; C07D243/14; C07D267/14; C07D279/16; C07D413/06
Domestic Patent References:
JP4321669A
JP8301848A
JP7002800A
JP4154765A
JP2003513082A
JP200739466A
Other References:
J. MED. CHEM.,1996年,39(18),3547-3555
Attorney, Agent or Firm:
Takashima Ichi