Title:
グルココルチコイドレセプターのための非ステロイド性リガンド、その組成物および使用
Document Type and Number:
Japanese Patent JP4745609
Kind Code:
B2
Abstract:
The invention provides non-steroidal ligands for the glucocorticoid receptor, methods for making non-steroidal ligands of the glucocorticoid receptor, compositions of non-steroidal ligands of the glucocorticoid receptor and methods of using non-steroidal ligands and compositions of non-steroidal ligands of the glucocorticoid receptor for treating or preventing diseases (e.g., obesity, diabetes, depression, neurodegeneration or an inflammatory disease) associated with glucocorticoid binding to the glucocorticoid receptor.
More Like This:
Inventors:
Scanlan, Thomas, S.
Shah, Niresh
Shah, Niresh
Application Number:
JP2003561595A
Publication Date:
August 10, 2011
Filing Date:
January 22, 2003
Export Citation:
Assignee:
The Regents of The University of California
International Classes:
C07D231/54; A61K31/415; A61K31/416; A61K31/42; A61K31/423; A61K31/425; A61P3/04; A61P3/10; A61P5/44; A61P5/46; A61P25/22; A61P25/24; A61P25/28; A61P29/00; C07D275/06; C07D317/72; C07D327/10; C07D339/06; C07D403/06; C07D409/06
Foreign References:
| EP0102404A1 | ||||
| DE1169442A | ||||
| GB1071124B | ||||
| US3135743 | ||||
| GB934574B |
Other References:
Journal of Medicinal Chemistry ,1993年,36(22),pp.3278-3285
Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry,1999年,38B(7),pp.847-849
Planta Medica ,1999年,65(8),pp.778-779
薬学雑誌,1973年,93(3),pp.296-299
Journal of Organic Chemistry ,1962年,vol.27,pp.2800-2807
Tetrahedron Letters ,1994年,35(36),pp.6643-6646
Steroids,1992年,57(7),pp.306-312
Journal of Steroid Biochemistry,1990年,36(1-2),pp.153-174
Journal of Organic Chemistry ,1980年,45(14),pp.2741-2746
Journal of the Chemical Society [Section] D: Chemical Communications ,1971年,vol.5,pp.233-234
Journal of the Chemical Society [Section] C: Organic ,1969年,vol.14,pp.1937-1939
Chemical & Pharmaceutical Bulletin ,1968年,16(8),pp.1487-1497
Canadian Journal of Chemistry ,1963年,41(9),pp.2294-2298
Journal of Medicinal Chemistry ,2000年,43(22),pp.4233-4246
Journal of Medicinal Chemistry,2000年,43(9),pp.1866-1877
Biological & Pharmaceutical Bulletin ,1993年,16(2) ,pp.142-145
Life Sciences ,1992年,50(12),pp.891-897
Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry,1999年,38B(7),pp.847-849
Planta Medica ,1999年,65(8),pp.778-779
薬学雑誌,1973年,93(3),pp.296-299
Journal of Organic Chemistry ,1962年,vol.27,pp.2800-2807
Tetrahedron Letters ,1994年,35(36),pp.6643-6646
Steroids,1992年,57(7),pp.306-312
Journal of Steroid Biochemistry,1990年,36(1-2),pp.153-174
Journal of Organic Chemistry ,1980年,45(14),pp.2741-2746
Journal of the Chemical Society [Section] D: Chemical Communications ,1971年,vol.5,pp.233-234
Journal of the Chemical Society [Section] C: Organic ,1969年,vol.14,pp.1937-1939
Chemical & Pharmaceutical Bulletin ,1968年,16(8),pp.1487-1497
Canadian Journal of Chemistry ,1963年,41(9),pp.2294-2298
Journal of Medicinal Chemistry ,2000年,43(22),pp.4233-4246
Journal of Medicinal Chemistry,2000年,43(9),pp.1866-1877
Biological & Pharmaceutical Bulletin ,1993年,16(2) ,pp.142-145
Life Sciences ,1992年,50(12),pp.891-897
Attorney, Agent or Firm:
Atsushi Nakajima
Kato Kazunori
Katsuichi Nishimoto
Kato Kazunori
Katsuichi Nishimoto