Title:
NOVEL ALPHAAAMINOPHENYLACETIC ACID DERIVATIVE
Document Type and Number:
Japanese Patent JPS5533476
Kind Code:
A
Abstract:
1. Alpha-Aminophenylacetic acid derivatives of the general formula see diagramm : EP0011092,P18,F1 in which R**1 represents hydroxy or alkoxy with 1 to 4 carbon atoms, R**2 represents hydrogen, alkyl with 1 to 4 carbon atoms, trifluoromethyl or halogen, R**3 and R**4 are identical or different and in each case represent hydrogen, allyl or alkyl with up to 4 carbon atoms, the alkyl radicals being optionally substituted by amino, cyano or alkoxy with 1 to 2 carbon atoms or R**3 and R**4 together with the nitrogen atom form a 5-membered to 7-membered aliphatic ring, which can optionally be saturated or unsaturated and which can contain one oxygen atom, one sulphur atom, one SO grouping, one SO2 grouping or one N-R''' grouping, wherein R''' represents hydrogen, alkyl with 1 to 2 carbon atoms or methoxyethyl,or together with the nitrogen atom form a triacolyl radical. R**5 represents hydrogen or alkyl with 1 to 4 carbon atoms and R**6 represents hydrogen or alkyl with 1 to 2 carbon atoms, and pharmacologically acceptable salts thereof, for use in the treatment of inflammatory diseases.
Inventors:
GUNTAA SHIYUMITSUTO
BORUFUGANKU OPITSU
HAIREDEIN YAKOBI
BORUFUGANKU OPITSU
HAIREDEIN YAKOBI
Application Number:
JP10512679A
Publication Date:
March 08, 1980
Filing Date:
August 20, 1979
Export Citation:
Assignee:
BAYER AG
International Classes:
A61K31/165; A61K31/195; A61K31/215; A61K31/40; A61K31/41; A61K31/415; A61K31/445; A61K31/50; C07C67/00; C07C227/00; C07C227/18; C07C227/24; C07C229/42; C07C231/00; C07C231/02; C07C233/47; C07C237/20; C07C237/22; C07C253/00; C07C255/58; C07C255/60; C07C313/00; C07C323/63; C07D233/34; C07D233/36; C07D233/38; C07D233/76; C07D241/04; C07D249/06; C07D249/08; C07D295/14; C07D295/155; C07D295/205; (IPC1-7): A61K31/165; A61K31/195; A61K31/215; A61K31/41; C07C101/447; C07C103/28; C07C103/52; C07C103/76; C07C121/52; C07C149/32; C07D233/32; C07D249/06; C07D295/14