Title:
PHARMACEUTICAL COMPOSITION
Document Type and Number:
Japanese Patent JP2014015456
Kind Code:
A
Abstract:
To provide a pharmaceutical composition which contains as an active ingredient a consecutive aromacyclic compound which has an inhibitory action on diacylglycerol acyltransferase 1 that is an enzyme catalyzing a reaction from diacylglycerol to triglyceride and is useful for diseases associated with obesity.
Provided is a pharmaceutical composition containing as an active ingredient a consecutive aromacyclic compound, a representative example of which is 2,2-dimethyl-3-(4-{5-[5-(trifluoromethyl)-1H-imidazol-2-yl]pyridin-2-yl}phenoxy)propanoic acid represented by the following formula.
Inventors:
SAKURAI OSAMU
SARUTA KUNIO
HAYASHI NORIMITSU
GOI TAKASHI
MOROKUMA KENJI
TSUJIJIMA SHUICHI
SAWAMOTO HIROAKI
SHITAMA HIROAKI
IMASHIRO RITSUO
SARUTA KUNIO
HAYASHI NORIMITSU
GOI TAKASHI
MOROKUMA KENJI
TSUJIJIMA SHUICHI
SAWAMOTO HIROAKI
SHITAMA HIROAKI
IMASHIRO RITSUO
Application Number:
JP2013125519A
Publication Date:
January 30, 2014
Filing Date:
June 14, 2013
Export Citation:
Assignee:
MITSUBISHI TANABE PHARMA CORP
International Classes:
A61K31/4164; A61K31/4439; A61K31/444; A61K31/497; A61K31/501; A61K31/506; A61P1/16; A61P1/18; A61P3/04; A61P3/06; A61P3/10; A61P9/00; A61P9/10; A61P9/12; A61P11/00; A61P19/02; A61P43/00; C07D233/64; C07D401/04; C07D401/10; C07D401/14; C07D403/04; C07D403/10; C07D405/14
Domestic Patent References:
JP2007502862A | 2007-02-15 | |||
JP2009505962A | 2009-02-12 | |||
JP2013545719A | 2013-12-26 | |||
JP2007502862A | 2007-02-15 | |||
JP2009505962A | 2009-02-12 |
Foreign References:
WO2000078726A1 | 2000-12-28 | |||
WO2000078726A1 | 2000-12-28 |
Attorney, Agent or Firm:
Patent business corporation Tsukuni
Hajime Tsukuni
Yasuo Yanagibashi
Satoko Ito
Keiko Ozawa
Yoko Tanaka
Kurino Yuriko
Hajime Tsukuni
Yasuo Yanagibashi
Satoko Ito
Keiko Ozawa
Yoko Tanaka
Kurino Yuriko