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Title:
PHARMACEUTICAL COMPOSITION
Document Type and Number:
Japanese Patent JP2014015456
Kind Code:
A
Abstract:

To provide a pharmaceutical composition which contains as an active ingredient a consecutive aromacyclic compound which has an inhibitory action on diacylglycerol acyltransferase 1 that is an enzyme catalyzing a reaction from diacylglycerol to triglyceride and is useful for diseases associated with obesity.

Provided is a pharmaceutical composition containing as an active ingredient a consecutive aromacyclic compound, a representative example of which is 2,2-dimethyl-3-(4-{5-[5-(trifluoromethyl)-1H-imidazol-2-yl]pyridin-2-yl}phenoxy)propanoic acid represented by the following formula.


Inventors:
SAKURAI OSAMU
SARUTA KUNIO
HAYASHI NORIMITSU
GOI TAKASHI
MOROKUMA KENJI
TSUJIJIMA SHUICHI
SAWAMOTO HIROAKI
SHITAMA HIROAKI
IMASHIRO RITSUO
Application Number:
JP2013125519A
Publication Date:
January 30, 2014
Filing Date:
June 14, 2013
Export Citation:
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Assignee:
MITSUBISHI TANABE PHARMA CORP
International Classes:
A61K31/4164; A61K31/4439; A61K31/444; A61K31/497; A61K31/501; A61K31/506; A61P1/16; A61P1/18; A61P3/04; A61P3/06; A61P3/10; A61P9/00; A61P9/10; A61P9/12; A61P11/00; A61P19/02; A61P43/00; C07D233/64; C07D401/04; C07D401/10; C07D401/14; C07D403/04; C07D403/10; C07D405/14
Domestic Patent References:
JP2007502862A2007-02-15
JP2009505962A2009-02-12
JP2013545719A2013-12-26
JP2007502862A2007-02-15
JP2009505962A2009-02-12
Foreign References:
WO2000078726A12000-12-28
WO2000078726A12000-12-28
Attorney, Agent or Firm:
Patent business corporation Tsukuni
Hajime Tsukuni
Yasuo Yanagibashi
Satoko Ito
Keiko Ozawa
Yoko Tanaka
Kurino Yuriko