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Title:
PROSTAGLANDIN ANALOGUES,THEIR PREPARATION, AND PHARMACEUTICAL COMPOSIT IONS CONTAINING THE SAME AS ACTIVE INGREDIENT
Document Type and Number:
Japanese Patent JPS5227750
Kind Code:
A
Abstract:

PURPOSE: Prostaglandin analogues of formula I (Z is formula II, C=0; X is ethylene,cis-vinylene; Y is ethylene, trans-vinylene; R1 is H, 1W12C aliphatic alkyl), clathrates compounds thereof in cyclodextrin, or when R1 is H, nontoxic salts thereof. For example, 16-methylene-16-phenylthio-17,18,19,20-tetranor-prostaglandin F2α Me ester.


Inventors:
HAYASHI MASAKI
KOORI SEIJI
SHIMOJI KATSUICHI
Application Number:
JP10023076A
Publication Date:
March 02, 1977
Filing Date:
August 24, 1976
Export Citation:
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Assignee:
ONO PHARMACEUTICAL CO
International Classes:
A61K31/23; A61K31/20; A61K31/70; A61P43/00; C07C67/00; C07C401/00; C07C405/00; C08B37/16; (IPC1-7): A61K31/20; A61K31/23; A61K31/70; C07C177/00; C13L1/10



 
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