Title:
ピリジノン／ピラジノン、その作製方法、および使用方法
Document Type and Number:
Japanese Patent JP5841602
Kind Code:
B2
Abstract:
Pyridone and pyrazinone compounds of Formula I including stereoisomers, tautomers, and pharmaceutically acceptable salts thereof, useful for inhibiting Btk kinase, and for treating immune disorders such as inflammation mediated by Btk kinase. Methods of using compounds of Formula I for in vitro, in situ, and in vivo diagnosis, and treatment of such disorders in mammalian cells, or associated pathological conditions, are disclosed.
Inventors:
Kuri, Kevin S.
One, Xiao Jin
Young, Wendy Bee.
One, Xiao Jin
Young, Wendy Bee.
Application Number:
JP2013527279A
Publication Date:
January 13, 2016
Filing Date:
August 31, 2011
Export Citation:
Assignee:
Gilead Connecticut,Inc.
International Classes:
C07D401/14; A61K31/4439; A61K31/444; A61K31/496; A61K31/497; A61K31/4985; A61K31/501; A61K31/506; A61K31/5377; A61K31/5383; A61K31/542; A61K45/00; A61P1/04; A61P3/00; A61P7/00; A61P9/00; A61P11/06; A61P17/00; A61P17/06; A61P19/02; A61P25/00; A61P29/00; A61P31/12; A61P35/00; A61P35/02; A61P37/02; A61P37/06; A61P37/08; A61P43/00; C07D403/10; C07D403/14; C07D487/04; C07D495/04; C07D513/04; C07D519/00
Foreign References:
| WO2009053269A1 | ||||
| WO2009039397A1 | ||||
| WO2010100070A1 | ||||
| WO2010000633A1 | ||||
| WO2011140488A1 | ||||
| WO2010056875A1 |
Attorney, Agent or Firm:
Kiyoaki Takita
Nakamura Narumi
Iwasakizaki Ario
Nakamura Narumi
Iwasakizaki Ario