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Title:
PGDS阻害剤としてのピリミジンアミド化合物
Document Type and Number:
Japanese Patent JP5452925
Kind Code:
B2
Abstract:
This invention is directed to a compound of formula (I): wherein R1, R2, R3 and L1 are as defined herein, a pharmaceutical composition comprising the compound, and the use of the compound to treat allergic and/or inflammatory disorders, particularly disorders such as allergic rhinitis, asthma and/or chronic obstructive pulmonary disease (COPD).

Inventors:
Susan Sea Aldas
John Jiki Zean
Zinki Lou
Lian mar
Run Mu
Harry rundle manson
Jeffrey Stephen Sabor
Sukantini Tulai Ratnam
Christopher Lauren Van Dussen
Application Number:
JP2008534664A
Publication Date:
March 26, 2014
Filing Date:
October 04, 2006
Export Citation:
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Assignee:
Aventis Pharmaceuticals Incorporated
International Classes:
C07D401/04; A61K31/505; A61K31/506; A61K31/5377; A61K31/662; A61P11/00; A61P11/02; A61P11/06; A61P29/00; A61P37/08; C07D239/28; C07D403/12; C07D405/12; C07D417/12; C07F9/6512; C07D401/12; C07D401/14; C07D413/12; C07D413/14
Domestic Patent References:
JP3112985A
JP2002003370A
Foreign References:
WO2004072069A1
WO2005032493A1
US20050165028
Other References:
STN International,2-Phenylpyrimidine-5-carboxylic acid N-(3-trifluoromethylphenyl)amide,file REGISTRY [online],2005年2月15日掲載,[平成24年4月25日検索],CAS Registry No. 831240-98-3
Attorney, Agent or Firm:
Junji Yuda
Shoji Miwa
Noriyuki Takebayashi
Chika Takagi



 
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