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Title:
(R)-α-(2,3-ジメトキシフェニル)-1-[2-(4-フルオロフェニル)エチル]-4-ピペリジンメタノールの製造方法
Document Type and Number:
Japanese Patent JP4511723
Kind Code:
B2
Abstract:
The present invention provides various processes for the preparation of (R)-±-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol. These processes may be characterized by the following scheme:

Inventors:
Alan Gee Veena
Edward Dee Dougs
Jonathan Sea Evans
Hans-Wolfram Fleming
Gerard Guilamo
Robert A. Hawthorn
Thomas Ha A Hilpert
James E Hit
Qi-Shin Earl King
Johannes En Kuku
Frederik M. Larskoviks
John Earl Leffler
Alexey El Margolin
Sharon Kay Minish
Thomas Tea Autile
Lean Gee Rajuski
Marvin Jay Zack
Paul F Skartetti
Sandra Kay Stalls-Dan
Alonzo El Tigner
Ian A. Tomlinson
Application Number:
JP2000535626A
Publication Date:
July 28, 2010
Filing Date:
March 11, 1999
Export Citation:
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Assignee:
Aventis Holdings, Inc.
Sanofi-Aventis Deutschland Gesellschaft Mitt Beschlenktel Haftung
International Classes:
C07D211/22; A61K9/20; A61K31/4409; A61K31/445; A61K47/04; A61K47/12; A61K47/26; A61K47/38; A61P1/14; A61P7/02; A61P9/06; A61P9/08; A61P9/10; A61P21/00; A61P25/00; A61P25/18; A61P25/22; C07B57/00; C07B61/00; C07D211/32; C07D213/00; C07D213/30; C07D213/50
Domestic Patent References:
JP5507482A
Attorney, Agent or Firm:
Junji Yuda
Shoji Miwa
Noriyuki Takebayashi
Chika Takagi
Kosuke Nishimura