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Title:
RETROVIRAL PROTEASE-INHIBITING COMPOUND
Document Type and Number:
Japanese Patent JP2006232845
Kind Code:
A
Abstract:

To provide an HIV protease inhibitor useful for treating or preventing AIDS.

The retroviral protease-inhibiting compound is represented by general formula (A). Preferably, in the formula, R1 is a thiazolyl or oxazolyl which may be substituted; n is 1; R2 is hydrogen; R3 is a 1-4C alkyl; R4 and R4a are each phenyl; R6 is hydrogen; R7 is thiazolyl, oxazolyl or the like; and Z is O.


Inventors:
KEMPF DALE J
NORBECK DANIEL W
SHAM HING L
CHEN ZUAO
THOMAS J SOOUIN
DANIEL S RENO
HAIGHT ANTHONY R
ARTHUR J COOPER
Application Number:
JP2006103462A
Publication Date:
September 07, 2006
Filing Date:
April 04, 2006
Export Citation:
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Assignee:
ABBOTT LAB
International Classes:
C07D263/32; C07D275/02; A61K31/395; A61K31/415; A61K31/4164; A61K31/42; A61K31/421; A61K31/422; A61K31/425; A61K31/426; A61K31/427; A61K31/535; A61K31/5375; A61K31/5377; A61K31/54; A61K45/06; A61P31/12; A61P31/18; A61P35/00; A61P35/02; A61P37/04; A61P43/00; C07C33/46; C07C43/164; C07C43/174; C07C43/205; C07C43/215; C07C43/23; C07C43/30; C07C43/315; C07C45/00; C07C45/29; C07C45/56; C07C45/62; C07C45/67; C07C45/74; C07C53/134; C07C69/34; C07C69/65; C07C69/732; C07C211/27; C07C215/18; C07C215/20; C07C215/28; C07C229/08; C07C229/26; C07C229/34; C07C233/36; C07C233/40; C07C235/10; C07C235/12; C07C235/34; C07C235/78; C07C237/10; C07C237/20; C07C237/22; C07C239/10; C07C239/18; C07C239/20; C07C247/10; C07C251/40; C07C271/20; C07C271/22; C07C271/34; C07C275/16; C07C275/24; C07C311/03; C07C311/13; C07C311/18; C07C317/10; C07C317/28; C07C317/44; C07C323/12; C07C323/25; C07C381/00; C07D213/26; C07D213/30; C07D213/34; C07D213/40; C07D213/54; C07D213/56; C07D213/61; C07D213/75; C07D233/54; C07D233/84; C07D235/14; C07D235/16; C07D239/26; C07D241/12; C07D261/06; C07D261/08; C07D263/24; C07D263/30; C07D263/48; C07D265/30; C07D277/20; C07D277/22; C07D277/24; C07D277/26; C07D277/28; C07D277/30; C07D277/32; C07D277/34; C07D277/36; C07D277/40; C07D277/42; C07D277/56; C07D295/13; C07D295/205; C07D295/215; C07D303/36; C07D307/42; C07D333/16; C07D401/12; C07D413/12; C07D413/14; C07D417/12; C07D417/14; C07D521/00; C07F5/02; C07F5/04; C07K5/06; C07K5/065; A61K38/00; C07D235/10; C07D
Domestic Patent References:
JPH04308574A1992-10-30
JPH03207901A1991-09-11
JP2637847A
JP3812969A
JPH08505844A1996-06-25
Attorney, Agent or Firm:
Yoshio Kawaguchi