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Title:
セリンプロテアーゼインヒビター
Document Type and Number:
Japanese Patent JP2004503538
Kind Code:
A
Abstract:
Compounds of formula (I) where R5, R6a, each X, L, Cy and Lp are as defined in the specification, are tryptase inhibitors useful as antiinflammatory agents.

Inventors:
Sarah Elizabeth Lively
Bourdan Waskowitz
Martin James Harrison
Christopher Neil Farthing
Keith Michael Johnson
Application Number:
JP2002510448A
Publication Date:
February 05, 2004
Filing Date:
June 12, 2001
Export Citation:
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Assignee:
TULARIK LIMITED
International Classes:
C07D233/64; A61K31/166; A61K31/341; A61K31/343; A61K31/381; A61K31/405; A61K31/4172; A61K31/423; A61K31/426; A61K31/427; A61K31/428; A61K31/44; A61K31/445; A61K31/4465; A61K31/454; A61P1/00; A61P1/04; A61P1/16; A61P1/18; A61P7/02; A61P9/00; A61P9/10; A61P11/00; A61P11/02; A61P11/06; A61P11/08; A61P13/10; A61P15/00; A61P15/12; A61P17/00; A61P17/02; A61P17/04; A61P17/06; A61P19/02; A61P25/00; A61P25/06; A61P27/02; A61P29/00; A61P31/12; A61P35/00; A61P43/00; C07C237/42; C07C237/52; C07D209/08; C07D209/20; C07D211/34; C07D211/46; C07D211/60; C07D213/56; C07D213/61; C07D213/73; C07D233/54; C07D263/54; C07D273/00; C07D277/20; C07D277/30; C07D277/40; C07D277/46; C07D277/52; C07D277/68; C07D277/82; C07D307/54; C07D307/79; C07D307/81; C07D333/36; C07D333/60; C07D401/12; C07D417/12; (IPC1-7): C07C237/52; A61K31/166; A61K31/341; A61K31/343; A61K31/381; A61K31/405; A61K31/4172; A61K31/423; A61K31/426; A61K31/427; A61K31/428; A61K31/44; A61K31/445; A61K31/4465; A61K31/454; A61P1/00; A61P1/04; A61P1/16; A61P1/18; A61P9/00; A61P9/10; A61P11/00; A61P11/02; A61P11/06; A61P11/08; A61P13/10; A61P15/00; A61P15/12; A61P17/00; A61P17/02; A61P17/04; A61P17/06; A61P19/02; A61P25/00; A61P25/06; A61P27/02; A61P29/00; A61P31/12; A61P35/00; A61P43/00; C07D209/20; C07D211/34; C07D213/56; C07D213/73; C07D233/64; C07D263/54; C07D277/46; C07D277/52; C07D277/593; C07D277/82; C07D307/54; C07D307/81; C07D333/60; C07D401/12; C07D417/12
Domestic Patent References:
JP2004503547A2004-02-05
JP2004503532A2004-02-05
JP2003502314A2003-01-21
Foreign References:
WO1999026925A11999-06-03
WO1997037969A11997-10-16
Attorney, Agent or Firm:
Aoyama Aoi
Osamu Kawamiya
Kyousei Tamura
Hiromitsu Takayama