Title:
SUBSTITUTED 1*55CYLLOHEXADIENE CARBOXYLIC ACID DERIVATIVES
Document Type and Number:
Japanese Patent JPS54100349
Kind Code:
A
Abstract:
Compounds of the following general formula and salts thereof are irreversible inhibitors of gamma -aminobutyric acid transaminase: wherein R1 is hydrogen, alkylcarbonyl wherein the alkyl moiety has from 1 to 4 carbon atoms and is straight or branched, alkoxycarbonyl wherein the alkoxy moiety has from 1 to 4 carbon atoms and is straight or branched, the radical wherein R4 is hydrogen, a straight or branched alkyl group having from 1 to 4 carbon atoms, benzyl or p-hydroxybenzyl; R2 is hydroxy, a straight or branched alkoxy group of from 1 to 8 carbon atoms, the group -NR5R6 wherein each of R5 and R6 is hydrogen or a straight or branched alkyl group having from 1 to 4 carbon atoms, or wherein R7 is hydrogen, a straight or branched lower alkyl group of from 1 to 4 carbon atoms, benzyl or p-hydroxybenzyl; and R3 is hydrogen or bromine.
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Inventors:
BURIAN UORUTAA METOKARUFU
MISHIERU YUNKU
MISHIERU YUNKU
Application Number:
JP34079A
Publication Date:
August 08, 1979
Filing Date:
January 08, 1979
Export Citation:
Assignee:
MERRELL TORAUDE & CO
International Classes:
A61K31/00; A61K31/165; A61K31/19; A61K31/195; A61K31/215; A61K31/24; A61K31/27; A61P25/00; C07C61/22; A61K31/16; C07C67/00; C07C229/48; C07C231/00; C07C231/02; C07C233/52; C07C233/54; C07C237/04; C07C237/20; C07C237/24; C07C239/00; C07C271/24; C07C; (IPC1-7): A61K31/16; A61K31/19; A61K31/215; C07C99/00; C07C101/38; C07C102/00; C07C103/19; C07C103/46; C07C103/737; C07C125/04
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