Title:
置換4-アミノ-1-ベンジルピペリジン化合物
Document Type and Number:
Japanese Patent JP2007524641
Kind Code:
A
Abstract:
This invention provides 4-amino-1-benzylpiperidine and related compounds and pharmaceutically acceptable salts thereof which are useful as muscarinic receptor antagonists. This invention also provides pharmaceutical compositions containing such compounds; processes and intermediates useful for preparing such compounds; and methods for treating disease conditions mediated by muscarinic receptors, such as overactive bladder, irritable bowel syndrome, asthma and chronic obstructive pulmonary disease, using such compounds.
Inventors:
Mamen, masai
Wilson, Richard
Dunham, Sara
Hughes, Adam
Hasfeld, Craig
The, You Hua
Lee, lee
Mishki, Trevor
Sturgiers, Ioana
Ore, david
Wilson, Richard
Dunham, Sara
Hughes, Adam
Hasfeld, Craig
The, You Hua
Lee, lee
Mishki, Trevor
Sturgiers, Ioana
Ore, david
Application Number:
JP2006518963A
Publication Date:
August 30, 2007
Filing Date:
July 09, 2004
Export Citation:
Assignee:
Theravans, Incorporated
International Classes:
C07D401/06; A61K31/454; A61K31/5377; A61P1/00; A61P11/00; A61P11/06; A61P13/00; A61P13/10; A61P43/00; C07D401/12; C07D401/14; C07D405/14; C07D407/14
Domestic Patent References:
JP2003516391A | 2003-05-13 | |||
JPH04500521A | 1992-01-30 | |||
JPH04505927A | 1992-10-15 | |||
JPH05501554A | 1993-03-25 |
Foreign References:
WO2002056016A2 | 2002-07-18 | |||
WO2004041806A2 | 2004-05-21 | |||
WO2005003090A1 | 2005-01-13 |
Attorney, Agent or Firm:
Hidesaku Yamamoto
Takaaki Yasumura
Natsuki Morishita
Takaaki Yasumura
Natsuki Morishita