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Title:
置換4-アミノ-1-ベンジルピペリジン化合物
Document Type and Number:
Japanese Patent JP2007524641
Kind Code:
A
Abstract:
This invention provides 4-amino-1-benzylpiperidine and related compounds and pharmaceutically acceptable salts thereof which are useful as muscarinic receptor antagonists. This invention also provides pharmaceutical compositions containing such compounds; processes and intermediates useful for preparing such compounds; and methods for treating disease conditions mediated by muscarinic receptors, such as overactive bladder, irritable bowel syndrome, asthma and chronic obstructive pulmonary disease, using such compounds.

Inventors:
Mamen, masai
Wilson, Richard
Dunham, Sara
Hughes, Adam
Hasfeld, Craig
The, You Hua
Lee, lee
Mishki, Trevor
Sturgiers, Ioana
Ore, david
Application Number:
JP2006518963A
Publication Date:
August 30, 2007
Filing Date:
July 09, 2004
Export Citation:
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Assignee:
Theravans, Incorporated
International Classes:
C07D401/06; A61K31/454; A61K31/5377; A61P1/00; A61P11/00; A61P11/06; A61P13/00; A61P13/10; A61P43/00; C07D401/12; C07D401/14; C07D405/14; C07D407/14
Domestic Patent References:
JP2003516391A2003-05-13
JPH04500521A1992-01-30
JPH04505927A1992-10-15
JPH05501554A1993-03-25
Foreign References:
WO2002056016A22002-07-18
WO2004041806A22004-05-21
WO2005003090A12005-01-13
Attorney, Agent or Firm:
Hidesaku Yamamoto
Takaaki Yasumura
Natsuki Morishita