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Title:
IRAK4阻害剤としての置換インダゾール化合物
Document Type and Number:
Japanese Patent JP2017518348
Kind Code:
A
Abstract:
本発明は、式(I)の置換インダゾール化合物およびその薬学的に許容される塩、ならびにIRAK4を阻害するため、および/またはIRAK4により誘導される疾患または障害の治療のためのそれらの使用を提供する。

Inventors:
Gamadi, Ben Keatswar Lao
Samaji Dar, Santa
Application Number:
JP2016574004A
Publication Date:
July 06, 2017
Filing Date:
June 19, 2015
Export Citation:
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Assignee:
AURIGENE DISCOVERY TECHNOLOGIES LIMITED
International Classes:
C07D401/14; A61K31/437; A61K31/4439; A61K31/4453; A61K31/496; A61P1/02; A61P1/04; A61P1/16; A61P1/18; A61P3/04; A61P3/06; A61P5/00; A61P7/00; A61P7/02; A61P7/06; A61P9/12; A61P11/00; A61P11/02; A61P11/04; A61P11/06; A61P13/00; A61P13/08; A61P13/12; A61P17/00; A61P17/04; A61P17/06; A61P17/14; A61P19/00; A61P19/02; A61P19/08; A61P21/00; A61P21/04; A61P25/00; A61P25/04; A61P25/06; A61P27/02; A61P27/12; A61P29/00; A61P35/00; A61P35/02; A61P37/00; A61P37/02; A61P37/06; A61P37/08; A61P43/00; C07D413/14; C07D451/06; C07D471/04; C07D487/04
Domestic Patent References:
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Foreign References:
WO2013068458A12013-05-16
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Other References:
BIOORG. MED. CHEM., vol. 12, JPN6019005696, 2004, pages 2115 - 2137, ISSN: 0003980211
BIOORG. MED. CHEM. LETT., vol. 14, JPN6019005698, 2004, pages 6011 - 6016, ISSN: 0003980212
REGISTRY(STN)[ONLINE], JPN7019000449, 2011, ISSN: 0003980213
REGISTRY(STN)[ONLINE], JPN7019000450, 2014, ISSN: 0003980214
Attorney, Agent or Firm:
Yusuke Hiraki
Satoshi Fujita
Eiichi Arai
Natsuo Tanaka
Naoko Kikuta