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Patent Searching and Data


Title:
ヒストンデアセチラーゼの新規な阻害剤としての置換されたプロペニルピペラジン誘導体
Document Type and Number:
Japanese Patent JP5279268
Kind Code:
B2
Abstract:
This invention comprises the novel compounds of formula (I) wherein R1, R2, R3, R4 and X have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.

Inventors:
Van Brandt, Sven Franciscus Anna
Van Emmelen, Christoph
Anjibo, Patrick Rene
Marconet-Declan, Lawrence Francoise Bernadette
Artz, Janine
Application Number:
JP2007523072A
Publication Date:
September 04, 2013
Filing Date:
July 25, 2005
Export Citation:
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Assignee:
JANSSEN PHARMACEUTICA NAAMLOZE VENNOOTSCHAP
International Classes:
C07D213/82; A61K31/506; A61K31/5377; A61P17/06; A61P35/00; A61P43/00; C07D239/42; C07D403/12
Foreign References:
WO2003075929A1
Attorney, Agent or Firm:
Patent business corporation Odashima patent office