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Title:
SUBSTITUTED PYRAZOLYL COMPOUND FOR TREATING INFLAMMATION
Document Type and Number:
Japanese Patent JP2009029808
Kind Code:
A
Abstract:

To provide a substituted pyrazolyl derivative for treating cancer, inflammation and inflammation-associated disorders such as arthritis.

A compound having a structural formula expressed by figure is cited as an example. The compound is 1-{4-[(aminothio)peroxy]phenyl}-8-nitro-4,5-dihydro-1H-benzo[g]indazole-3-carboxamide.


Inventors:
BERGMANIS ARIJA A
BONAFOUX DOMINIQUE
CLARE MICHAEL
CRICH JOYCE Z
FLETCHER THERESA R
GENG LIFENG
HAGEN TIMOTHY J
HAMPER BRUCE C
HANSON GUNNAR J
HOUDEK STEPHEN C
HUANG HE
IULA DONNA M
KOSZYK FRANCIS J
LENNON PATRICK J
LIAO SHUYUAN
LIAO SUBO
METZ SUZANNE
MOHLER SCOTT B
NGUYEN MARIA
OBURN DAVID S
OWEN THOMAS J
PARTIS RICHARD A
SCATES ANGELA M
STEALEY MICHAEL A
TOLLEFSON MICHAEL B
VAZQUEZ MICHAEL L
WEIER RICHARD M
WOLFSON SERGE G
XU XIANGDONG
Application Number:
JP2008188020A
Publication Date:
February 12, 2009
Filing Date:
July 22, 2008
Export Citation:
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Assignee:
PHARMACIA CORP
International Classes:
C07D231/54; A61K31/416; A61K31/4178; A61K31/4245; A61K31/427; A61K31/433; A61K31/437; A61K31/4439; A61K31/444; A61K31/455; A61K31/4709; A61K31/4725; A61K31/496; A61K31/506; A61K31/5377; A61K31/551; A61P19/02; A61P25/04; A61P29/00; A61P35/00; C07D333/62; C07D401/04; C07D401/10; C07D401/12; C07D401/14; C07D403/10; C07D403/12; C07D405/04; C07D405/10; C07D405/12; C07D405/14; C07D409/12; C07D409/14; C07D413/12; C07D417/12; C07D417/14; C07D471/04
Attorney, Agent or Firm:
Junji Yuda
Shoji Miwa
Noriyuki Takebayashi
Chika Takagi