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Title:
オキシトシン拮抗薬としての置換トリアゾール誘導体
Document Type and Number:
Japanese Patent JP2007505888
Kind Code:
A
Abstract:
The present invention relates to a class of substituted 1,2,4-triazoles of formula (I) with activity as oxytocin antagonists, uses thereof, processes for the preparation thereof and compositions containing, said, inhibitors. These inhibitors have utility in a variety of therapeutic areas including sexual dysfunction, particularly premature ejaculation (P.E.).

Inventors:
Alan Daniel Brown
David Ellis
Christopher Ronald Smith
Application Number:
JP2006526721A
Publication Date:
March 15, 2007
Filing Date:
September 10, 2004
Export Citation:
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Assignee:
Pfizer Inc.
International Classes:
C07D249/08; A61K31/4196; A61K31/444; A61K31/497; A61K31/501; A61K31/506; A61P1/16; A61P5/10; A61P9/04; A61P9/12; A61P13/08; A61P15/00; A61P15/06; A61P15/10; A61P25/18; A61P27/02; C07D401/04; C07D401/14; C07D403/04; C07D403/14
Domestic Patent References:
JP2000063363A2000-02-29
Foreign References:
WO2003053437A12003-07-03
WO2001087855A12001-11-22
WO2001058880A12001-08-16
Attorney, Agent or Firm:
Chika Takagi
Junji Yuda
Shoji Miwa