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Title:
スルファモイル−アリールアミド及びＢ型肝炎の治療のための薬剤としてのその使用
Document Type and Number:
Japanese Patent JP2015533782
Kind Code:
A
Abstract:
式（Ｉ）のＨＢＶ複製の阻害薬であり、その立体化学異性体、並びに塩、水和物、溶媒和化合物を含み、式中、Ｂ、Ｒ１、Ｒ２及びＲ４は、本明細書に定義した通りの意味を有する。本発明はまた、前記化合物を製造する方法、これらを含む医薬組成物、及びＨＢＶ治療における単独での、又は他のＨＢＶ阻害薬と併用したその使用にも関する。【化１】

Inventors:
Van Dick, Cohen
Last, stephan, julian
Rhombu, Gale
Werschlen, Wim, Gaston
La Boisson, Pierre, Jean-Marie, Bernard
Application Number:
JP2015529007A
Publication Date:
November 26, 2015
Filing Date:
August 28, 2013
Export Citation:
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Assignee:
Janssen Sciences Ireland Ireland
International Classes:
C07C311/16; A61K31/18; A61K31/337; A61K31/34; A61K31/341; A61K31/351; A61K31/397; A61K31/40; A61K31/4168; A61K31/426; A61K31/438; A61K31/44; A61K31/4402; A61K31/4453; A61K31/4468; A61K31/45; A61K31/495; A61K31/5375; A61K31/55; A61P31/12; A61P31/20; C07C311/17; C07C311/20; C07C311/51; C07D205/02; C07D207/12; C07D207/26; C07D211/56; C07D211/58; C07D211/76; C07D211/96; C07D213/42; C07D213/81; C07D233/84; C07D277/56; C07D295/04; C07D295/12; C07D295/22; C07D305/08; C07D307/22; C07D307/64; C07D309/14; C07D333/34; C07D333/48; C07D491/107; C07D491/113; C07D493/08
Domestic Patent References:
JP2010535172A2010-11-18
JP2015531773A2015-11-05
JP2011513250A2011-04-28
Foreign References:
WO2010123139A12010-10-28
US20050239833A12005-10-27
US20050221272A12005-10-06
WO2009018219A22009-02-05
CN102206172A2011-10-05
WO2013096744A12013-06-27
WO2013006394A12013-01-10
WO2013130703A22013-09-06
US20100016310A12010-01-21
WO2009131065A12009-10-29
US20090259044A12009-10-15
Other References:
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Attorney, Agent or Firm:
Hiroshi Kobayashi
Junko Kobayashi
Norio Omori
Yasuhito Suzuki



 
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