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Title:
【発明の名称】オキサチエピノ[6,5-b]ジヒドロピリジン類、並びに関連組成物および方法
Document Type and Number:
Japanese Patent JP2003504373
Kind Code:
A
Abstract:
This invention provides novel oxathiepino[6,5-b]dihydropyridines. These compounds are useful as calcium channel antagonists with cardiovascular, antiasthmatic and antibronchoconstriction activity. Thus, this invention also provides pharmaceutical compositions, as well as methods, for preventing and treating disorders such as hypersensitivity, allergy, asthma, bronchospasm, dysmenorrhea, esophageal spasm, glaucoma, premature labor, urinary tract disorders, gastrointestinal motility disorders and cardiovascular disorders.

Inventors:
Dotsudo, Jiyoung H
Henry The Ames Earl
Rupert, Kenneth See
Barrington, The Ames El
Hall, Daniel A.
Application Number:
JP2001509733A
Publication Date:
February 04, 2003
Filing Date:
June 23, 2000
Export Citation:
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Assignee:
Ortho-McNeill Pharmacy Incorporated
International Classes:
A61K31/4365; A61P1/06; A61P1/14; A61P9/00; A61P9/04; A61P9/10; A61P9/12; A61P11/00; A61P11/06; A61P11/08; A61P13/04; A61P15/00; A61P15/06; A61P25/02; A61P27/06; A61P37/08; C07D495/04; C07D497/04; C07D221/00; C07D327/00; (IPC1-7): C07D497/04; A61K31/4365; A61P1/06; A61P1/14; A61P9/04; A61P9/10; A61P9/12; A61P11/06; A61P11/08; A61P13/04; A61P15/00; A61P15/06; A61P25/02; A61P27/06; A61P37/08
Attorney, Agent or Firm:
Heiyoshi Odashima