Title:
【発明の名称】PLA▲下2▼阻害剤としてのエステル類およびアミド類
Document Type and Number:
Japanese Patent JP3353301
Kind Code:
B2
Abstract:
The present invention relates to a novel fatty acid derivative of the following formula: wherein R1 is acyl group; R2 is acyl(lower)alkyl; R3 is hydrogen, aryl(lower)alkyl, etc; R4 is acyl(lower)alkyl; and X is -O-, [wherein R5 is lower alkyl, etc]; and a pharmaceutically acceptable salt thereof, which is useful as a medicament; the processes for the preparation of said fatty acid derivative or a salt thereof; a pharmaceutical composition comprising said fatty acid derivative or a pharmaceutically acceptable salt thereof; etc.
Inventors:
Naoki Fukami
Seiji Yoshimura
Keisuke Imai
Heiji Emi
Seiji Yoshimura
Keisuke Imai
Heiji Emi
Application Number:
JP50653897A
Publication Date:
December 03, 2002
Filing Date:
July 18, 1996
Export Citation:
Assignee:
Fujisawa Pharmaceutical Co., Ltd.
International Classes:
A61K31/16; A61K31/165; A61K31/215; A61K31/34; A61K31/343; A61K31/40; A61K31/403; A61K31/404; A61K31/44; A61K31/4427; A61K31/443; A61K31/47; A61K31/472; A61P9/00; A61P29/00; A61P37/00; A61P37/08; A61P43/00; C07C235/34; C07C237/22; C07C269/06; C07C271/22; C07D209/42; C07D215/48; C07D215/54; C07D217/22; C07D217/26; C07D233/54; C07D233/66; C07D307/80; C07D401/06; C07D401/12; C07D405/12; (IPC1-7): C07C235/34; A61K31/16; A61K31/165; A61K31/215; A61K31/34; A61K31/40; A61K31/44; A61K31/47; A61P9/00; A61P29/00; A61P37/00; A61P37/08; A61P43/00; C07C237/22; C07C271/22; C07D209/42; C07D215/48; C07D215/54; C07D217/22; C07D307/80; C07D401/06; C07D401/12; C07D405/12
Domestic Patent References:
| JP625195A | ||||
| JP7112970A | ||||
| JP6505497A | ||||
| JP2500030A | ||||
| JP9508363A |
Other References:
【文献】国際公開93/6127(WO,A1)
【文献】国際公開93/21211(WO,A1)
【文献】国際公開93/21211(WO,A1)
Attorney, Agent or Firm:
Eiji Tabuse