Title:
【発明の名称】ピラゾロ〔4,3-c〕ピリジン類、その製造方法およびそれを含有するセロトニン再摂取阻害剤
Document Type and Number:
Japanese Patent JP2656211
Kind Code:
B2
Abstract:
The invention relates to compounds of the frmula wherein Ar is or pyridyl; R1 is H,-(CH2)pNR2R3, R2 is hydrogen or loweralkyl; R3 is hydrogen or loweralkyl; R4 is hydrogen or loweralkyl; X and Y are independently halogen, trifluoromethyl, nitro, loweralkyl, loweralkoxy or hydroxy; n is 0, 1, 2 or 3; m is 0, 1 or 2; p and q are independently 2, 3 or 4; or a pharmaceutically acceptable addition salt and/or hydrate thereof, or where applicable, a geometric or optical isomer or racemic mixture thereof. This invention also relates to a process for making the compounds and to pharmaceutical compositions, and to their use as serotonin reuptake inhibitors.
Inventors:
GUREGORII MAIKURU SHATSUTSUKE
KEBIN JEIMUZU KATSUPURUZU
JON DEITSUKU TOMAA ZAFUOOSU
KEBIN JEIMUZU KATSUPURUZU
JON DEITSUKU TOMAA ZAFUOOSU
Application Number:
JP26515893A
Publication Date:
September 24, 1997
Filing Date:
October 22, 1993
Export Citation:
Assignee:
HEKISUTO MARION RUSERU INC
International Classes:
A61K31/44; A61K31/445; A61P25/00; A61P25/18; A61P25/24; A61K31/435; A61P25/26; C07D471/04; (IPC1-7): C07D471/04; A61K31/435; A61K31/44; A61K31/445
Other References:
ＣＨＥＭＩＣＡＬ ＡＢＳＴＲＡＣＴＳ 第１０８巻要約番号１１１４４８（１９８８）ＢＵＬＬ．ＣＨＥＭ．ＳＯＣ．ＪＡＰ．，４４〜３！（１９７１）Ｐ．８５８−８５９
Attorney, Agent or Firm:
Chika Takagi (2 outside)