Title:
【発明の名称】レトロウイルスプロテアーゼ抑制化合物
Document Type and Number:
Japanese Patent JP2963910
Kind Code:
B2
Abstract:
A retroviral protease inhibiting compound of the formula A - X - B or a pharmaceutically acceptable salt, prodrug or ester thereof, wherein X is a linking group; A is (1) substituted amino, (2) substituted carbonyl, (3) functionalized imino, (4) functionalized alkyl, (5) functionalized acyl, (6) functionalized heterocyclic or (7) functionalized (heterocyclic)alkyl; and B is (1) substituted carbonyl independently defined as herein, (2) substituted amino independently defined as herein, (3) functionalized imino independently defined as herein, (4) functionalized alkyl independently defined as herein, (5) functionalized acyl independently defined as herein, (6) functionalized heterocyclic independently defined as herein or (7) functionalized (heterocyclic)alkyl independently defined as herein. o
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Inventors:
DEIRU JEI KENPU
DANIERU DABURYU NOOBETSUKU
JON DABURYU ERIKUSON
HIN REUN SHAMU
RIN EMU KODAKOBI
YAKOBU JEI PURATSUTONAA
DANIERU DABURYU NOOBETSUKU
JON DABURYU ERIKUSON
HIN REUN SHAMU
RIN EMU KODAKOBI
YAKOBU JEI PURATSUTONAA
Application Number:
JP13368490A
Publication Date:
October 18, 1999
Filing Date:
May 23, 1990
Export Citation:
Assignee:
ABOTSUTO LAB
International Classes:
C07D295/18; A61K31/00; A61K31/10; A61K31/12; A61K31/135; A61K31/15; A61K31/165; A61K31/195; A61K31/335; A61K31/40; A61K31/415; A61K31/425; A61K31/44; A61K31/445; A61K31/47; A61K31/495; A61K31/535; A61K31/54; A61K38/00; A61P31/12; A61P37/04; C07C31/125; C07C33/18; C07C33/26; C07C33/46; C07C39/12; C07C43/164; C07C43/174; C07C43/205; C07C43/215; C07C43/23; C07C43/30; C07C43/313; C07C43/315; C07C45/00; C07C45/29; C07C45/56; C07C45/59; C07C45/62; C07C45/67; C07C45/74; C07C49/04; C07C49/12; C07C49/17; C07C49/175; C07C49/20; C07C49/215; C07C49/233; C07C49/24; C07C49/255; C07C53/134; C07C69/34; C07C69/65; C07C69/732; C07C211/27; C07C215/06; C07C215/18; C07C215/20; C07C215/28; C07C217/04; C07C225/06; C07C229/08; C07C229/26; C07C229/34; C07C233/35; C07C233/36; C07C233/40; C07C233/78; C07C235/10; C07C235/12; C07C235/34; C07C235/78; C07C237/04; C07C237/10; C07C237/20; C07C237/22; C07C239/08; C07C239/10; C07C239/18; C07C239/20; C07C247/10; C07C251/40; C07C271/20; C07C271/22; C07C271/34; C07C275/00; C07C275/16; C07C275/24; C07C311/03; C07C311/05; C07C311/06; C07C311/13; C07C311/18; C07C317/10; C07C317/28; C07C317/44; C07C323/11; C07C323/12; C07C323/25; C07C323/41; C07C323/60; C07C381/00; C07D207/06; C07D207/08; C07D207/12; C07D207/16; C07D207/24; C07D209/42; C07D211/22; C07D211/54; C07D211/62; C07D211/96; C07D213/30; C07D213/40; C07D213/42; C07D213/55; C07D213/56; C07D213/70; C07D213/81; C07D213/82; C07D215/16; C07D217/14; C07D217/16; C07D217/26; C07D231/10; C07D233/60; C07D233/61; C07D233/84; C07D239/38; C07D263/06; C07D263/32; C07D277/24; C07D277/28; C07D277/36; C07D277/42; C07D277/56; C07D279/12; C07D295/088; C07D295/14; C07D295/15; C07D295/155; C07D295/185; C07D295/20; C07D295/205; C07D295/215; C07D295/22; C07D295/26; C07D303/04; C07D303/22; C07D303/36; C07D303/48; C07D305/14; C07D307/42; C07D317/12; C07D413/12; C07D417/12; C07D487/04; C07D521/00; C07F7/02; C07F9/30; C07F9/32; C07F9/53; C07K5/02; C07K5/04; C07K5/06; C07K5/062; C07K5/078; (IPC1-7): C07C215/06; A61K31/00; A61K31/10; A61K31/12; A61K31/135; A61K31/15; A61K31/165; A61K31/195; A61K31/335; A61K31/40; A61K31/415; A61K31/425; A61K31/44; A61K31/445; A61K31/47; A61K31/495; A61K31/535; A61K31/54; C07C31/125; C07C33/18; C07C33/26; C07C33/46; C07C39/12; C07C43/23; C07C43/30; C07C49/04; C07C49/12; C07C49/17; C07C49/175; C07C49/20; C07C49/24; C07C49/255; C07C217/04; C07C225/06; C07C233/35; C07C233/78; C07C237/04; C07C237/20; C07C237/22; C07C239/08; C07C275/00; C07C311/03; C07C317/10; C07C317/28; C07C317/44; C07C323/11; C07C323/41; C07C323/60; C07D207/06; C07D207/08; C07D207/12; C07D209/42; C07D211/22; C07D211/96; C07D213/30; C07D213/55; C07D217/14; C07D217/16; C07D217/26; C07D231/10; C07D233/60; C07D233/84; C07D277/24; C07D277/28; C07D279/12; C07D295/14; C07D295/18; C07D295/20; C07D295/22; C07D303/48; C07D305/14; C07D307/42; C07D317/12; C07D487/04; C07F7/02; C07F9/30; C07K5/062
Attorney, Agent or Firm:
Aoyama Ryo (1 person outside)
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