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Title:
【発明の名称】プロゲステロンレセプタ結合剤として用いるための置換2-アリールイミノ複素環類およびそれを含有する組成物
Document Type and Number:
Japanese Patent JP2002534517
Kind Code:
A
Abstract:
This invention relates to 2-arylimino heterocycles, including 2-arylimino-1, 3-thiazolidines, 2-arylimino-2, 3, 4, 5-tetrahydro-1, 3-thiazines, 2-arylimino-1, 3-thiazolidin-4-ones, 2-arylimino-1, 3-thiazolidin-5-ones, and 2-arylimino-1, 3-oxazolidines, and their use in modulating progesterone receptor mediated processes, and pharmaceutical compositions for use in such therapies.

Inventors:
Brian Earle, Dixon
Bagi, Sed Em
Brennan, Katherine Earl
Brittelli, David Earl
Baroque, William H
Chiang, Jinshiang
Corbye, William El
Robert Dally
Ji Young Sung, Jeffrey S
Klunder, Harold See Yi
Lathrop, William F
Riu, paying
Maceor, Carroll Ann
Redman, Anico M
Scott, William J.A.
Woolburns, Claus
Wollanine, Donald J. Ray
Application Number:
JP2000593599A
Publication Date:
October 15, 2002
Filing Date:
December 14, 1999
Export Citation:
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Assignee:
BAYER CORPORATION
International Classes:
A61K31/4164; A61K31/421; A61K31/423; A61K31/425; A61K31/426; A61K31/427; A61K31/428; A61K31/429; A61K31/437; A61K31/54; A61K31/55; A61P5/00; A61P5/24; A61P9/00; A61P9/10; A61P13/00; A61P15/00; A61P15/04; A61P15/08; A61P15/10; A61P15/16; A61P15/18; A61P17/00; A61P19/00; A61P19/10; A61P25/00; A61P25/24; A61P25/28; A61P35/00; A61P41/00; C07D263/28; C07D263/52; C07D233/42; C07D277/18; C07D277/20; C07D277/42; C07D277/54; C07D277/60; C07D279/06; C07D281/02; C07D417/06; C07D417/12; C07D513/04; C07D513/10; A61K; A61P; C07D; (IPC1-7): C07D277/18; A61K31/4164; A61K31/421; A61K31/425; A61K31/427; A61K31/428; A61K31/429; A61K31/437; A61K31/54; A61P5/00; A61P5/24; A61P9/10; A61P13/00; A61P15/00; A61P15/04; A61P15/08; A61P15/10; A61P15/16; A61P17/00; A61P19/00; A61P19/10; A61P25/00; A61P25/24; A61P25/28; A61P35/00; A61P41/00; C07D233/42; C07D263/28; C07D277/42; C07D277/60; C07D279/06; C07D417/06; C07D417/12; C07D513/04; C07D513/10
Attorney, Agent or Firm:
Heiyoshi Odashima