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Title:
【発明の名称】新規の置換α-ヒドロキシカルボン酸誘導体、その製造方法およびエンドセリンレセプターアンタゴニストとしての使用
Document Type and Number:
Japanese Patent JP2001523671
Kind Code:
A
Abstract:
The present invention relates to carboxylic acid derivatives of the formula Ithe substituents having the meanings explained in the description, preparation and use as endothelin receptor antagonists.

Inventors:
Wilhelm Amberg
Rolf Jansen
Heinz Hillen
Stephan Helgen Radar
Manfred Rashack
Liliane Unger
Application Number:
JP2000521084A
Publication Date:
November 27, 2001
Filing Date:
November 04, 1998
Export Citation:
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Assignee:
BASF Akchen Gezel Shaft
International Classes:
A61K31/41; A61K31/415; A61K31/4164; A61K31/42; A61K31/421; A61K31/422; A61K31/4245; A61K31/425; A61K31/426; A61K31/427; A61K31/428; A61K31/433; A61P9/04; A61P9/08; A61P9/10; A61P9/12; A61P11/06; A61P13/08; A61P13/12; A61P35/00; A61P43/00; C07D231/20; C07D233/70; C07D261/12; C07D263/38; C07D271/06; C07D271/10; C07D273/01; C07D275/02; C07D275/03; C07D277/20; C07D277/32; C07D277/34; C07D277/60; C07D277/68; C07D285/00; C07D285/08; C07D285/12; C07D291/04; C07D249/12; C07D413/12; C07D417/12; (IPC1-7): A61K31/425; A61K31/41; A61K31/415; A61K31/4164; A61K31/42; A61K31/421; A61K31/422; A61K31/4245; A61K31/426; A61K31/427; A61K31/428; A61K31/433; A61P9/04; A61P9/08; A61P9/10; A61P9/12; A61P11/06; A61P13/08; A61P13/12; A61P35/00; A61P43/00; C07D231/20; C07D233/70; C07D249/12; C07D261/12; C07D263/38; C07D271/06; C07D271/10; C07D273/01; C07D275/03; C07D277/34; C07D277/60; C07D277/68; C07D285/00; C07D285/08; C07D285/12; C07D291/04; C07D413/12; C07D417/12
Attorney, Agent or Firm:
Toshio Yano (4 outside)