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Title:
骨髄異形成症候群の処置
Document Type and Number:
Japanese Patent JP2016525532
Kind Code:
A
Abstract:
本発明は、骨髄異形成症候群(MDS)の処置のための、ボラセルチブ又は薬学的に許容されるその塩若しくはその水和物の使用に関する。

Inventors:
Rudolph, Dorsia
Tauve, Tillman
Application Number:
JP2016528536A
Publication Date:
August 25, 2016
Filing Date:
July 24, 2014
Export Citation:
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Assignee:
Boehringer Ingelheim International GmbH
International Classes:
C07D475/00; A61K31/519; A61P7/00; A61P35/02; A61P43/00
Domestic Patent References:
JP2009515852A2009-04-16
JP2008509949A2008-04-03
JP2015540794A2013-11-01
Foreign References:
WO2012072505A12012-06-07
WO2014071109A12014-05-08
Other References:
EUR. J. CANCER, vol. 48, JPN6018021821, 2012, pages 179 - 186, ISSN: 0003816591
MAHESH SEETHARAM ET AL: "Treatment of higher risk myelodysplastic syndrome patients unresponsive to hypomethylatin agents wit", LEUKEMIA RESEARCH, vol. 36(1), JPN6018021822, 2012, pages 98 - 103, ISSN: 0003816592
BERG T; BUG G; OTTMANN O G; STREBHARDT K: "POLO-LIKE KINASES IN AML", EXPERT OPINION ON INVESTIGATIONAL DRUGS, vol. VOL:21 NR:8, JPN5016008344, August 2012 (2012-08-01), pages 1069 - 1074, ISSN: 0003816593
LEONIDAS BENETATOS; AGGELIKI DASOULA; ELEFTHERIA HATZIMICHAEL; NELOFER SYED ET AL: "POLO-LIKE KINASE 2 (SNK/PLK2) IS A NOVEL EPIGENETICALLY REGULATED GENE IN ACUTE MYELOID 以下備考", ANNALS OF HEMATOLOGY, vol. VOL:90 NR:9, JPN5016008345, September 2011 (2011-09-01), DE, pages 1037 - 1045, ISSN: 0003816594
CHRISTOPH D C; SCHULER M: "POLO-LIKE KINASE 1 INHIBITORS IN MONO- AND COMBINATION THERAPIES: A 以下備考", EXPERT REVIEW OF ANTICANCER THERAPY, vol. VOL:11 NR:7, JPN5016008346, July 2011 (2011-07-01), GB, pages 1115 - 1130, ISSN: 0003816595
Attorney, Agent or Firm:
Patent business corporation Tsukuni